Synthesis and insecticidal activity of N-cyano 2-(substituted amino) ethyl methyl sulfoximine derivatives

被引：0

作者：

Yu, Haibo ^{[1
]}

Qin, Zhenfang ^{[1
]}

Dai, Hong ^{[1
]}

Zhang, Xin ^{[1
]}

Qin, Xue ^{[1
]}

Wang, Tingting ^{[1
]}

Fang, Jianxin ^{[1
]}

机构：

[1] Nankai Univ, Res Inst Elementoorgan Chem, State Key Lab Elementoorgan Chem, Tianjin 300071, Peoples R China

来源：

ARKIVOC | 2008年

基金：

中国国家自然科学基金;

关键词：

Sulfoximine derivatives; synthesis; insecticidal activity; peach aphid;

D O I：

10.3998/ark.5550190.0009.g10

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The N-cyano 2-(substituted amino) ethyl methyl sulfoximine derivatives are a new chemical family of neonicotinoids. Nine alkyl sulfoximine derivatives were designed and synthesized. The synthesized compounds were identified by H-1 NMR, C-13 NMR, IR, and elemental analysis. The preliminary bioassays indicated that some of them showed moderate insecticidal activities against Myzus persicae. The relationship between structure and biological activity was also discussed.

引用

页码：99 / 109

页数：11

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