Synthesis and novel structure-activity relationships of potent sansalvamide A derivatives

被引：30
|
作者：
Otrubova, K
Styers, TJ
Pan, PS
Rodriguez, R
McGuire, KL
McAlpine, SR
机构：
[1] San Diego State Univ, Dept Chem & Biochem, San Diego, CA 92182 USA
[2] San Diego State Univ, Dept Biol, San Diego, CA 92182 USA
来源：
CHEMICAL COMMUNICATIONS | 2006年 / 09期
关键词：
D O I：
10.1039/b517434a
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Synthesis of twelve Sansalvamide A derivatives and their SAR against colon cancer (HT- 29).
引用
收藏
页码：1033 / 1034
页数：2
相关论文
共 50 条
  • [1] Synthesis and Structure-Activity Relationships of Novel Neocryptolepine Derivatives
    El-Gokha, Ahmed A.
    Boshta, Nader M.
    Hussein, Mona K. Abo
    El Sayed, Ibrahim El-T.
    CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2017, 33 (03) : 373 - 377
  • [2] Synthesis and structure-activity relationships of novel neocryptolepine derivatives
    Ahmed A. El-Gokha
    Nader M. Boshta
    Mona K. Abo Hussein
    Ibrahim El-T. El Sayed
    Chemical Research in Chinese Universities, 2017, 33 : 373 - 377
  • [3] Synthesis and structure-activity relationships of novel warfarin derivatives
    Gebauer, Markus
    BIOORGANIC & MEDICINAL CHEMISTRY, 2007, 15 (06) : 2414 - 2420
  • [4] Synthesis, pharmacological evaluation, and structure-activity relationships of benzopyran derivatives with potent SERM activity
    Amari, G
    Armani, E
    Ghirardi, S
    Delcanale, M
    Civelli, M
    Caruso, PL
    Galbiati, E
    Lipreri, M
    Rivara, S
    Lodola, A
    Mor, M
    BIOORGANIC & MEDICINAL CHEMISTRY, 2004, 12 (14) : 3763 - 3782
  • [5] Synthesis and structure-activity relationships of potent antitumor active quinoline and naphthyridine derivatives
    Srivastava, Sanjay K.
    Jha, Amrita
    Agarwal, Shiv K.
    Mukherjee, Rama
    Burman, Anand C.
    ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, 2007, 7 (06) : 685 - 709
  • [6] Synthesis, fugicidal activity and quantitative structure-activity relationships of novel flavanone derivatives
    Yang, GF
    Ding, Y
    Yang, HZ
    Wu, XJ
    CHEMICAL JOURNAL OF CHINESE UNIVERSITIES-CHINESE, 2004, 25 (01): : 71 - 75
  • [7] Structure-activity relationships of novel potent MurF inhibitors
    Gu, YG
    Florjancic, AS
    Clark, RF
    Zhang, TY
    Cooper, CS
    Anderson, DD
    Lerner, CG
    McCall, JO
    Cai, YN
    Black-Schaefer, CL
    Stamper, GF
    Hajduk, PJ
    Beutel, BA
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2004, 14 (01) : 267 - 270
  • [8] Synthesis of sansalvamide A derivatives: Novel templates as potent antitumor agents
    Singh, Erinprit K.
    Rodriguez, Rodrigo
    Styers, Thomas J.
    Pan, Po-Shen
    Pan, Chung-Mao
    Ravula, Suchitra
    Lapera, Stephanie
    Cajica, Julia
    Brown, Joseph D.
    Parry, Emily
    McAlpine, Shelli
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 233 : 569 - 569
  • [9] Novel potent neuropeptide YY5 receptor antagonists: Synthesis and structure-activity relationships of phenylpiperazine derivatives
    Takahashi, Toshiyuki
    Sakuraba, Aya
    Hirohashi, Tomoko
    Shibata, Takunobu
    Hirose, Masaaki
    Haga, Yuji
    Nonoshita, Katsumasa
    Kanno, Tetsuya
    Ito, Junko
    Iwaasa, Hisashi
    Kanatani, Akio
    Fukami, Takehiro
    Sato, Nagaaki
    BIOORGANIC & MEDICINAL CHEMISTRY, 2006, 14 (22) : 7501 - 7511
  • [10] Evaluation of Di-Sansalvamide A Derivatives: Synthesis, Structure-Activity Relationship, and Mechanism of Action
    Alexander, Leslie D.
    Sellers, Robert P.
    Davis, Melinda R.
    Ardi, Veronica C.
    Johnson, Victoria A.
    Vasko, Robert C.
    McAlpine, Shelli R.
    JOURNAL OF MEDICINAL CHEMISTRY, 2009, 52 (24) : 7927 - 7930
12345