Synthesis of glycoprotein inhibitory agents sinuxylamide A-E

被引:5
作者
Annapurna, K. [1 ]
Rao, K. Srinivasa [1 ]
Narsaiah, A. Venkat [1 ,2 ]
机构
[1] CSIR Indian Inst Chem Technol, Organ Synth Lab, Fluoroagrochem Dept, Hyderabad 500007, Telangana, India
[2] Acad Sci & Innovat Res AcSIR, CSIR HRDC Campus Postal Staff Coll Area Sect 19, Ghaziabad 201002, Uttar Pradesh, India
来源
INDIAN JOURNAL OF CHEMISTRY | 2022年 / 61卷 / 10期
关键词
L-Tyrosine; Amide; Etherification; Glycoprotein; Marine products;
D O I
10.56042/ijc.v61i10.64005
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Synthesis of naturally occurring Sinuxylamides A-E has been accomplished. Synthesis started from commercially available L-tyrosine. The key reactions involved in this synthesis are amide formation, Mitsunobu etherification and ester hydrolysis.
引用
收藏
页码:1039 / 1045
页数:7
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