A novel method for the racemization of 5-bromonicotine

被引：12

作者：

Bleicher, LS

Cosford, NDP

机构：

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1999年 / 64卷 / 14期

关键词：

D O I：

10.1021/jo990152g

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：5299 / 5300

页数：2

共 10 条

[1] TRANSFORMATIONS INVOLVING THE PYRROLIDINE RING OF NICOTINE [J].

ACHESON, RM ;

FERRIS, MJ ;

SINCLAIR, NM .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1980, (02) :579-585

[2] A practical and efficient synthesis of the selective neuronal acetylcholine-gated ion channel agonist (S)-(-)-5-ethynyl-3-(1-methyl-2-pyrrolidinyl)pyridine maleate (SIB-1508Y) [J].

Bleicher, LS ;

Cosford, NDP ;

Herbaut, A ;

McCallum, JS ;

McDonald, IA .

JOURNAL OF ORGANIC CHEMISTRY, 1998, 63 (04) :1109-1118

[3] A CONVENIENT METHOD FOR THE PREPARATION OF RACEMIC NICOTINE [J].

BOWMAN, ER ;

MCKENNIS, H ;

MARTIN, BR .

SYNTHETIC COMMUNICATIONS, 1982, 12 (11) :871-879

[4] OPTICAL RESOLUTION BY DIRECT CRYSTALLIZATION OF ENANTIOMER MIXTURES [J].

COLLET, A ;

BRIENNE, MJ ;

JACQUES, J .

CHEMICAL REVIEWS, 1980, 80 (03) :215-230

[5] Controlled racemization of optically active organic compounds: Prospects for asymmetric transformation [J].

Ebbers, EJ ;

Ariaans, GJA ;

Houbiers, JPM ;

Bruggink, A ;

Zwanenburg, B .

TETRAHEDRON, 1997, 53 (28) :9417-9476

[6] Neuronal nicotinic acetylcholine receptors as targets for drug discovery [J].

Holladay, MW ;

Dart, MJ ;

Lynch, JK .

JOURNAL OF MEDICINAL CHEMISTRY, 1997, 40 (26) :4169-4194

[7]

HOOTELE C, 1974, CHIMIA, V28, P665

[8] Facile pyridoxal-catalyzed racemization of nornicotine and related compounds [J].

Jacob, P .

JOURNAL OF ORGANIC CHEMISTRY, 1996, 61 (09) :2916-2917

[9] CRYSTALLIZATION-INDUCED ASYMMETRIC TRANSFORMATION - STEREOSPECIFIC SYNTHESIS OF A POTENT PERIPHERAL CCK ANTAGONIST [J].

REIDER, PJ ;

DAVIS, P ;

HUGHES, DL ;

GRABOWSKI, EJJ .

JOURNAL OF ORGANIC CHEMISTRY, 1987, 52 (05) :955-957

[10]

TSUJINO Y, 1982, HETEROCYCLES, V19, P2151

← 1 →