A one pot microwave assisted synthesis of 3-acyl-2,4-dihydroxyquinoline followed by synthesis of 7-methyldibenzo[c,f][2,7]naphthyridin-6(5H)-ones via three routes

被引：0

作者：

Pitchai, P. ^{[1
,2
,3
]}

Uvarani, C. ^{[2
]}

Gengan, R. M. ^{[3
]}

Mohan, P. S. ^{[2
]}

机构：

[1] Govt Arts Coll Autonomous, PG & Res Dept Chem, Kumbakonam 612001, India

[2] Bharathiar Univ, Dept Chem, Sch Chem Sci, Coimbatore 641046, Tamil Nadu, India

[3] Durban Univ Technol, Dept Chem, ZA-4001 Durban, South Africa

来源：

INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 2013年 / 52卷 / 06期

基金：

新加坡国家研究基金会;

关键词：

Microwave; eco-friendly; photochemical cyclization; naphthyridines; 3-acyl-2,4-dihydroxyquinoline; PHOTOCHEMICAL-REACTIONS; DERIVATIVES; INHIBITORS; ALKALOIDS; AGENTS;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An easy one pot microwave assisted synthesis of 3-acyl-2,4-dihydroxyquinoline from simple precursors followed by convenient synthesis of novel and potential HIV integrase inhibitors 7-methyldibenzo[c,f][2,7]naphthyridin-6(5H)-ones has been achieved through three different routes. Mild reaction conditions and good yields are obtained by applying microwave and photochemical techniques.

引用

页码：776 / 786

页数：11

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