Solvent-free synthesis of new heteryl β-ketosulfones

被引：9

作者：

Guravaiah, Nalajam ^{[1
]}

Rao, Vedula Rajeswar ^{[1
]}

机构：

[1] Natl Inst Technol, Dept Chem, Warangal 506021, Andhra Pradesh, India

来源：

JOURNAL OF CHEMICAL RESEARCH | 2009年 / 02期

关键词：

3-(2-bromoacetyl)coumarin; sodiumarenesulfinate; beta-ketosulfones; solvent-free synthesis; KETO-SULFONES; COUMARIN DERIVATIVES; GAMMA-AMINO; ACETYLENES; DESULFONYLATION; SULFOXIDES; CHLORIDES; EFFICIENT; WATER;

D O I：

10.3184/030823409X401745

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A novel efficient method for the coupling of sulfinic acid salts and alpha-halo ketones is described. A variety of heteryl beta-ketosulfones have been formed in an excellent yields at room temperature under solvent-free conditions.

引用

页码：87 / 89

页数：3

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