High-resolution X-ray crystallography reveals precise binding interactions between human nonpancreatic secreted phospholipase A(2) and a highly potent inhibitor (FPL67047XX)

被引：36
|
作者：
Cha, SS
Lee, D
Adams, J
Kurdyla, JT
Jones, CS
Marshall, LA
Bolognese, B
AbdelMeguid, SS
Oh, BH
机构：
[1] SMITHKLINE BEECHAM PHARMACEUT, DEPT MACROMOL SCI, KING OF PRUSSIA, PA 19406 USA
[2] SMITHKLINE BEECHAM PHARMACEUT, DEPT MED CHEM, KING OF PRUSSIA, PA 19406 USA
[3] SMITHKLINE BEECHAM PHARMACEUT, DEPT BIOCHEM, KING OF PRUSSIA, PA 19406 USA
[4] SMITHKLINE BEECHAM PHARMACEUT, DEPT INFLAMMAT & RESP PHARMACOL, KING OF PRUSSIA, PA 19406 USA
[5] POHANG UNIV SCI & TECHNOL, DEPT LIFE SCI, KYUNGBUK 790784, SOUTH KOREA
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 1996年 / 39卷 / 20期
关键词：
D O I：
10.1021/jm960502g
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
[No abstract available]
引用
收藏
页码：3878 / 3881
页数：4
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