共 72 条
[71]
Challenges in the development of mGluR5 positive allosteric modulators: The discovery of CPPHA
[J].
Zhao, Zhijian
;
Wisnoski, David D.
;
O'Brien, Julie A.
;
Lemaire, Wei
;
Williams, David L., Jr.
;
Jacobson, Marlene A.
;
Wittman, Marion
;
Ha, Sookhee N.
;
Schaffhauser, Herve
;
Sur, Cyrille
;
Pettibone, Doug J.
;
Duggan, Mark E.
;
Conn, P. Jeffrey
;
Hartman, George D.
;
Lindsley, Craig W.
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
2007, 17 (05)
:1386-1391

Zhao, Zhijian
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Wisnoski, David D.
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

O'Brien, Julie A.
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Lemaire, Wei
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Williams, David L., Jr.
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Jacobson, Marlene A.
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Wittman, Marion
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Ha, Sookhee N.
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Schaffhauser, Herve
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Sur, Cyrille
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Pettibone, Doug J.
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Duggan, Mark E.
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Conn, P. Jeffrey
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Hartman, George D.
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA

Lindsley, Craig W.
论文数: 0 引用数: 0
h-index: 0
机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA
[72]
Discovery of N-Aryl Piperazines as Selective mGluR5 Potentiators with Improved In Vivo Utility
[J].
Zhou, Ya
;
Manka, Jason T.
;
Rodriguez, Alice L.
;
Weaver, C. David
;
Days, Emily L.
;
Vinson, Paige N.
;
Jadhav, Satyawan
;
Hermann, Elizabeth J.
;
Jones, Carrie K.
;
Conn, P. Jeffrey
;
Lindsley, Craig W.
;
Stauffer, Shaun R.
.
ACS MEDICINAL CHEMISTRY LETTERS,
2010, 1 (08)
:433-438

Zhou, Ya
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA
Vanderbilt Univ, Med Ctr, Vanderbilt Program Drug Discovery, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA

Manka, Jason T.
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA
Vanderbilt Univ, Med Ctr, Vanderbilt Program Drug Discovery, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA

Rodriguez, Alice L.
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA
Vanderbilt Univ, Med Ctr, Vanderbilt Program Drug Discovery, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA

Weaver, C. David
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA
Vanderbilt Univ, Med Ctr, Vanderbilt Program Drug Discovery, Nashville, TN 37232 USA
Vanderbilt Inst Chem Biol, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA

Days, Emily L.
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Vanderbilt Program Drug Discovery, Nashville, TN 37232 USA
Vanderbilt Inst Chem Biol, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA

Vinson, Paige N.
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA
Vanderbilt Univ, Med Ctr, Vanderbilt Program Drug Discovery, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA

Jadhav, Satyawan
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA
Vanderbilt Univ, Med Ctr, Vanderbilt Program Drug Discovery, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA

Hermann, Elizabeth J.
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA
Vanderbilt Univ, Med Ctr, Vanderbilt Program Drug Discovery, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA

Jones, Carrie K.
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA
Vanderbilt Univ, Med Ctr, Vanderbilt Program Drug Discovery, Nashville, TN 37232 USA
Tennessee Valley Healthcare Syst, US Dept Vet Affairs, Nashville, TN 37212 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA

Conn, P. Jeffrey
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA
Vanderbilt Univ, Med Ctr, Vanderbilt Program Drug Discovery, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA

Lindsley, Craig W.
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA
Vanderbilt Univ, Med Ctr, Dept Chem, Nashville, TN 37232 USA
Vanderbilt Univ, Med Ctr, Vanderbilt Program Drug Discovery, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA

Stauffer, Shaun R.
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA
Vanderbilt Univ, Med Ctr, Vanderbilt Program Drug Discovery, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA