A novel accurate method of human protein tyrosine phosphatase 1B inhibitors high-throughput screening

被引:0
|
作者
Pang, Xiao-bin [1 ,2 ]
Xie, Xin-mei [1 ]
Zhao, Qing-hui [1 ]
Wang, Shou-bao [2 ,3 ]
Du, Guan-hua [2 ,3 ]
机构
[1] Henan Univ, Inst Pharmaceut, Kaifeng 475004, Peoples R China
[2] Chinese Acad Med Sci, Inst Mat Med, Natl Ctr Pharmaceut Screening, Beijing 100050, Peoples R China
[3] Peking Union Med Coll, Beijing 100050, Peoples R China
来源
ACTA PHARMACOLOGICA SINICA | 2013年 / 34卷
关键词
protein tyrosine phosphatase 1B; inhibitor; high-throughput screening; insulin receptor;
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
引用
收藏
页码:45 / 46
页数:2
相关论文
共 50 条
  • [31] Toward the identification of a reliable 3D-QSAR model for the protein tyrosine phosphatase 1B inhibitors
    Wang, Fangfang
    Zhou, Bo
    JOURNAL OF MOLECULAR STRUCTURE, 2018, 1158 : 75 - 87
  • [32] Phosphorylation and activation of protein tyrosine phosphatase (PTP) 1B by insulin receptor
    Dadke, S
    Kusari, A
    Kusari, J
    MOLECULAR AND CELLULAR BIOCHEMISTRY, 2001, 221 (1-2) : 147 - 154
  • [33] Phosphorylation and activation of protein tyrosine phosphatase (PTP) 1B by insulin receptor
    Shrikrishna Dadke
    Anasua Kusari
    Jyotirmoy Kusari
    Molecular and Cellular Biochemistry, 2001, 221 : 147 - 154
  • [34] Stearic Acid Serves as a Potent Inhibitor of Protein Tyrosine Phosphatase 1B
    Tsuchiya, Ayako
    Kanno, Takeshi
    Nishizaki, Tomoyuki
    CELLULAR PHYSIOLOGY AND BIOCHEMISTRY, 2013, 32 (05) : 1451 - 1459
  • [35] Analysis of in vitro interactions of protein tyrosine phosphatase 1B with insulin receptors
    Wang, XY
    Bergdahl, K
    Heijbel, A
    Liljebris, C
    Bleasdale, JE
    MOLECULAR AND CELLULAR ENDOCRINOLOGY, 2001, 173 (1-2) : 109 - 120
  • [36] Computational revelation of binding mechanisms of inhibitors to endocellular protein tyrosine phosphatase 1B using molecular dynamics simulations
    Yan, Fangfang
    Liu, Xinguo
    Zhang, Shaolong
    Su, Jing
    Zhang, Qinggang
    Chen, Jianzhong
    JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS, 2018, 36 (14): : 3636 - 3650
  • [37] 4-Quinolone-3-carboxylic acids as cell-permeable inhibitors of protein tyrosine phosphatase 1B
    Zhi, Ying
    Gao, Li-Xin
    Jin, Yi
    Tang, Chun-Lan
    Li, Jing-Ya
    Li, Jia
    Long, Ya-Qiu
    BIOORGANIC & MEDICINAL CHEMISTRY, 2014, 22 (14) : 3670 - 3683
  • [38] A novel high-throughput screening format to identify inhibitors of secreted acid sphingomyelinase
    Mintzer, RJ
    Appell, KC
    Cole, A
    Johns, A
    Pagila, R
    Polokoff, MA
    Tabas, I
    Snider, RM
    Meurer-Ogden, JA
    JOURNAL OF BIOMOLECULAR SCREENING, 2005, 10 (03) : 225 - 234
  • [39] Discovery of novel Leishmania major trypanothione synthetase inhibitors by high-throughput screening
    Phan, Trong-Nhat
    Park, Kyuho Paul
    Benitez, Diego
    Comini, Marcelo A.
    Shum, David
    No, Joo Hwan
    BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2022, 637 : 308 - 313
  • [40] Structural and molecular insights of protein tyrosine phosphatase 1B (PTP1B) and its inhibitors as anti-diabetic agents
    Paul, Abhik
    Sarkar, Arnab
    Banerjee, Tanmoy
    Maji, Avik
    Sarkar, Shrabanti
    Paul, Sourav
    Karmakar, Sanmoy
    Ghosh, Nilanjan
    Maity, Tapan Kumar
    JOURNAL OF MOLECULAR STRUCTURE, 2023, 1293