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- [42] Rational design of potent and selective VLA-4 inhibitors and their utility in the treatment of asthmaCURRENT TOPICS IN MEDICINAL CHEMISTRY, 2004, 4 (14) : 1497 - 1507Singh, J论文数: 0 引用数: 0 h-index: 0机构: Biogen Inc, Cambridge, MA 02142 USA Biogen Inc, Cambridge, MA 02142 USAAdams, S论文数: 0 引用数: 0 h-index: 0机构: Biogen Inc, Cambridge, MA 02142 USA Biogen Inc, Cambridge, MA 02142 USACarter, MB论文数: 0 引用数: 0 h-index: 0机构: Biogen Inc, Cambridge, MA 02142 USA Biogen Inc, Cambridge, MA 02142 USACuervo, H论文数: 0 引用数: 0 h-index: 0机构: Biogen Inc, Cambridge, MA 02142 USA Biogen Inc, Cambridge, MA 02142 USALee, WC论文数: 0 引用数: 0 h-index: 0机构: Biogen Inc, Cambridge, MA 02142 USA Biogen Inc, Cambridge, MA 02142 USALobb, RR论文数: 0 引用数: 0 h-index: 0机构: Biogen Inc, Cambridge, MA 02142 USA Biogen Inc, Cambridge, MA 02142 USAPepinsky, RB论文数: 0 引用数: 0 h-index: 0机构: Biogen Inc, Cambridge, MA 02142 USA Biogen Inc, Cambridge, MA 02142 USAPetter, R论文数: 0 引用数: 0 h-index: 0机构: Biogen Inc, Cambridge, MA 02142 USA Biogen Inc, Cambridge, MA 02142 USAScott, D论文数: 0 引用数: 0 h-index: 0机构: Biogen Inc, Cambridge, MA 02142 USA Biogen Inc, Cambridge, MA 02142 USA
- [43] Synthesis, characterization and evaluation of pro-drugs of VLA-4 antagonists (Vol 14, pg 1651, 2004)BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2004, 14 (21) : 5449 - 5449Huryn, DM论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USAAshwell, S论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USABaudy, R论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USADressen, DB论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USAGallaway, W论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USAGrant, FS论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USAKonradi, A论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USALey, RW论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USAPetusky, S论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USAPleiss, MA论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USASarantakis, D论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USASemko, CM论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USASherman, MM论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USATio, C论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USAZhang, L论文数: 0 引用数: 0 h-index: 0机构: Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USA
- [44] Discovery and evaluation of N-(triazin-1,3,5-yl) phenylalanine derivatives as VLA-4 integrin antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2002, 12 (12) : 1591 - 1594Porter, JR论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandArchibald, SC论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandBrown, JA论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandChilds, K论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandCritchley, D论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandHead, JC论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandHutchinson, B论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandParton, TAH论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandRobinson, MK论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandShock, A论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandWarrellow, GJ论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandZomaya, A论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, England
- [45] N-(pyrimidin-4-yl) and N-(pyridin-2-yl) phenylalanine derivatives as VLA-4 integrin antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2002, 12 (12) : 1595 - 1598Porter, JR论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandArchibald, SC论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandBrown, JA论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandChilds, K论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandCritchley, D论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandHead, JC论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandHutchinson, B论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandParton, TAH论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandRobinson, MK论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandShock, A论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandWarrellow, GJ论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, EnglandZomaya, A论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Slough SL1 4EN, Berks, England Celltech R&D Ltd, Slough SL1 4EN, Berks, England
- [46] Novel N,N-disubstituted amides that are highly potent VLA-4 antagonists.ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2000, 219 : U53 - U53Kassir, JM论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USAScott, IL论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USABiediger, RJ论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USAGrabbe, VO论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USAMarket, RV论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USARaju, BG论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USALin, SQ论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USAKogan, TP论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USAChen, Q论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USAHolland, GW论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USAMaxwell, DC论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USAVanderslice, P论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USAWest, H论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USADecker, ER论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USABourgoyne, A论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USATilton, R论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USAMunsch, CL论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USADixon, RAF论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Chem, Houston, TX 77030 USA
- [47] 4-(pyrrolidinyl)methoxybenzoic acid derivatives as a potent, orally active VLA-4 antagonistCHEMICAL & PHARMACEUTICAL BULLETIN, 2006, 54 (11) : 1515 - 1529Chiba, Jun论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanIimura, Shin论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanYoneda, Yoshiyuki论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanSugimoto, Yuichi论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanHoriuchi, Takao论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanMuro, Fumito论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanOchiai, Yuichi论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanOgasawara, Tomomi论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanTsubokawa, Masao论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanIigou, Yutaka论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanTakayama, Gensuke论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanTaira, Tomoe论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanTakata, Yoshimi论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanYokoyama, Mika论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanTakashi, Tohru论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanNakayama, Atsushi论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, JapanMachinaga, Nobuo论文数: 0 引用数: 0 h-index: 0机构: Daiichi Pharmaceut Co Ltd, Med Chem Res Lab, Edogawa Ku, Tokyo 1348630, Japan
- [48] SAR studies of the leucine portion of Bio-1050, a potent and selective nanomolar antagonist of the integrin vla-4 (alpha(4)beta(1)).ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1997, 213 : 76 - MEDIZimmerman, CN论文数: 0 引用数: 0 h-index: 0机构: BIOGEN INC,DEPT MED CHEM,CAMBRIDGE,MA 02142 BIOGEN INC,DEPT MED CHEM,CAMBRIDGE,MA 02142Lin, KC论文数: 0 引用数: 0 h-index: 0机构: BIOGEN INC,DEPT MED CHEM,CAMBRIDGE,MA 02142 BIOGEN INC,DEPT MED CHEM,CAMBRIDGE,MA 02142
- [49] Discovery of DW-908: An orally potent and exquisitely selective VLA-4 antagonistABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238Machinaga, Nobuo论文数: 0 引用数: 0 h-index: 0机构: DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, Japan DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, JapanIimura, Shin论文数: 0 引用数: 0 h-index: 0机构: DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, Japan DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, JapanSugimoto, Yuuichi论文数: 0 引用数: 0 h-index: 0机构: DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, Japan DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, JapanYoneda, Yoshiyuki论文数: 0 引用数: 0 h-index: 0机构: DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, Japan DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, JapanChiba, Jun论文数: 0 引用数: 0 h-index: 0机构: DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, Japan DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, JapanWatanabe, Toshiyuki论文数: 0 引用数: 0 h-index: 0机构: DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, Japan DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, JapanMuro, Fumihito论文数: 0 引用数: 0 h-index: 0机构: DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, Japan DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, JapanSetoguchi, Masaki论文数: 0 引用数: 0 h-index: 0机构: DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, Japan DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, JapanNakayama, Atsushi论文数: 0 引用数: 0 h-index: 0机构: DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, Japan DAIICHI SANKYO CO LTD, Med Chem Res Labs 2, Edogawa Ku, Tokyo 1348630, Japan
- [50] TBC3486: Novel, highly potent, and selective VLA-4 antagonist.ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2000, 219 : U4 - U4Holland, GW论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAKassir, JM论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAScott, IL论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USABiediger, RJ论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USARen, K论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USARaju, BG论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAGrabbe, VO论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAMarket, RV论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USALin, SQ论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAKeller, KM论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAKogan, TP论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAKrudy, GA论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAChen, Q论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAMaxwell, DC论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAYou, TJ论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAVanderslice, P论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAWest, H论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USADecker, ER论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USABourgoyne, A论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USATilton, R论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USAMunsch, CL论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USADixon, RAF论文数: 0 引用数: 0 h-index: 0机构: Texas Biotechnol Corp, Houston, TX 77030 USA Texas Biotechnol Corp, Houston, TX 77030 USA