Synthesis of Unsaturated α-Acyloxybenzothiazoleamides via the Passerini Three-Component Reaction

被引：0

作者：

Sheikholeslami-Farahani, Fatemeh ^{[1
]}

Shahvelayati, Ashraf S. ^{[2
]}

机构：

[1] Islamic Azad Univ, Dept Chem, Firoozkooh Branch, Firoozkooh, Iran

[2] Islamic Azad Univ, Dept Chem, Shahr E Ray Branch, Tehran, Iran

来源：

COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING | 2013年 / 16卷 / 09期

关键词：

2-Aminobenzothiazole; maleic anhydride; passerini reaction; solvent-free media; MULTICOMPONENT REACTIONS; ALKYL ISOCYANIDES; CHEMISTRY; ACID; COMPONENT; UGI;

D O I：

暂无

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

4-Benzothiazol-2-ylamino-4-oxo-2-butenoic acid, prepared from reaction of 2-aminobenzothiazole and maleic anhydride, are used as an acid component in Passerini three-component reaction, under solvent-free media, to produce unsaturated alpha-benzothiazole acyloxyamides in good yields.

引用

页码：726 / 730

页数：5

共 24 条

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