NOVEL ONE-POT SYNTHESIS OF AZIRIDINES CARRYING SYDNONE MOIETY AND THEIR BIOLOGICAL STUDIES

被引：15

作者：

Hegde, Jyothi C. ^{[1
]}

Girish, K. S. ^{[1
]}

Adhikari, Adithya ^{[1
]}

Kalluraya, Balakrishna ^{[1
]}

机构：

[1] Mangalore Univ, Dept Studies Chem, Mangalagangthri, Karnataka, India

来源：

SYNTHETIC COMMUNICATIONS | 2013年 / 43卷 / 02期

关键词：

Aziridine; biological activity; one-pot synthesis; sydnone derivatives; DERIVATIVES; EPOXIDES;

D O I：

10.1080/00397911.2011.599102

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A novel series of 5-(3-arylsydnon-4-yl)-7-aryl-1,4-diazabicyclo[4,1,0]hept-4-enes 3a-l were prepared in a one-pot synthesis by the reaction of 2,3-dibromo-1-(3-arylsydnon-4-yl)-3-arylpropan-1-one 1a-l and 1,2-diaminoethane. The newly synthesized compounds were screened for their antibacterial and antifungal activity.

引用

页码：301 / 308

页数：8

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