Palladium-catalyzed decarboxylative C2-acylation of indoles with α-oxocarboxylic acids

被引：99
作者：
Pan, Changduo [1 ,2 ]
Jin, Hongming [1 ]
Liu, Xu [1 ]
Cheng, Yixiang [1 ]
Zhu, Chengjian [1 ,3 ]
机构：
[1] Nanjing Univ, Sch Chem & Chem Engn, State Key Lab Coordinat Chem, Nanjing 210093, Jiangsu, Peoples R China
[2] Wenzhou Inst Ind & Sci, Wenzhou 325000, Peoples R China
[3] Shanghai Inst Organ Chem, State Key Lab Organometall Chem, Shanghai 200032, Peoples R China
来源：
CHEMICAL COMMUNICATIONS | 2013年 / 49卷 / 28期
基金：
中国国家自然科学基金; 高等学校博士学科点专项科研基金;
关键词：
H BOND ACYLATION; OXIDATIVE ORTHO-ACYLATION; O-METHYL OXIMES; DIRECT ALKYNYLATION; C3; ALKENYLATION; ACETANILIDES; ALDEHYDES; CYANATION; FUNCTIONALIZATION; HETEROARENES;
D O I：
10.1039/c3cc40709h
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A palladium-catalyzed decarboxylative C2-acylation of indoles with alpha-oxocarboxylic acids was achieved. This protocol represents a novel and complementary approach to 2-aroylindoles.
引用
收藏
页码：2933 / 2935
页数：3
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