Synthesis of new 1-substituted 4-perfluoroalkyl tetrazol-5-ones

被引：22

作者：

Mekni, Nejib ^{[1
]}

Baklouti, Ahmed ^{[1
]}

机构：

[1] Fac Sci Tunis, Dept Chem, Lab Struct Organ Chem, Tunis 2092, Tunisia

来源：

JOURNAL OF FLUORINE CHEMISTRY | 2008年 / 129卷 / 11期

关键词：

1,4-Tetrazol-5-one; 1,3-Dipolar cycloaddition; Perfluoroalkyl azide; Isocyanate;

D O I：

10.1016/j.jfluchem.2008.06.019

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

1,3-Dipolar cycloaddition of perfluoroalkyl ethyle azides 1 with isocyanates 2 afforded 1-perfluoroalkyl-4-(n-Bu, phenyl or mesitylsulfonyl) tetrazol-5-ones 3 in good yields. The use of perfluoroalkyl ethyl azides extends the reaction to the less reactive n-butyl isocyanate. (c) 2008 Elsevier B.V. All rights reserved.

引用

页码：1073 / 1075

页数：3

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