Design, synthesis, and evaluation of potent and selective inhibitors of mono-(ADP-ribosyl) transferases, PARP10 and PARP14

被引:0
|
作者
Holechek, Jacob [2 ]
Lease, Robert [2 ]
Thorsell, Ann-Gerd [1 ]
Grant, Ryan [2 ]
Keen, Abby [2 ]
Karlberg, Tobias [1 ]
Schuler, Herwig [1 ]
Ferraris, Dana [2 ]
机构
[1] Karolinska Inst, Stockholm, Sweden
[2] McDaniel Coll, Chem, Westminster, MD USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
51
引用
收藏
页数:1
相关论文
共 33 条
  • [31] Design, synthesis, and biological evaluation of 2H-7-oxa-1,2-diaza-benzo[de]anthracen-3-one derivatives as potent PARP-1 inhibitors
    Xu, Weizheng
    Wilcoxen, Keith
    Zhang, Jie
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238
  • [32] Design, synthesis, and evaluation of aza-peptide Michael acceptors as selective and potent inhibitors of caspases-2, -3, -6, -7, -8, -9, and -10
    Ekici, Özlem Dogan
    Li, Zhao Zhao
    Campbell, Amy J.
    James, Karen Ellis
    Asgian, Juliana L.
    Mikolajczyk, Jowita
    Salvesen, Guy S.
    Ganesan, Rajkumar
    Jelakovic, Stjepan
    Gruetter, Markus G.
    Powers, James C.
    JOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (19) : 5728 - 5749
  • [33] Design and synthesis of poly(ADP-ribose)polymerase-1 (PARP-1) inhibitors.: Part 3:: In vitro evaluation of 1,3,4,5-tetrahydro-benzo[c][1,6] and [c][1,7]-naphthyridin-6-ones
    Ferraris, D
    Ficco, RP
    Pahutski, T
    Lautar, S
    Huang, S
    Zhang, J
    Kalish, V
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2003, 13 (15) : 2513 - 2518