Synthesis of (1H)-3,4-dihydropyrrolo[2,1-c][1,4]oxazin-1-one derivatives

被引:0
作者
Fu, DC [1 ]
Yu, H [1 ]
Zhang, SF [1 ]
机构
[1] Shenyang Pharmaceut Univ, Shenyang 110016, Peoples R China
关键词
(1H)-3,4-dihydropyrrolo[2,1-c][1,4]oxazin-1-; synthesis;
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
In search of new anti-inflammatory and analgesic agents, (1H)-3,4-dihydro- pyrrolo [2,1-c][1,4]oxazin-1-one (3) and its acyl derivatives were designed and prepared. compound 3 was prepared by treatment of methyl 1-(2-bromoethyl) pyrrole-2-carboxy late with silver oxide and its derivatives were obtained by Friedel-Cralles reaction. Nine of 6-acyl derivatives of compound 3 were prepared.
引用
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页码:1051 / 1054
页数:4
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