A concise and diversity-oriented strategy for the synthesis of benzofurans and indoles via Ugi and Diels-Alder reactions

被引：75
作者：
Lu, K
Luo, TP
Xiang, Z
You, ZJ
Fathi, R [1 ]
Chen, JH
Yang, Z
机构：
[1] Peking Univ, Key Lab Bioorgan Chem, Beijing 100871, Peoples R China
[2] Peking Univ, Coll Chem, Mol Engn Minist Educ, State Key Lab Nat & Biomimet Drugs,Sch Pharmaceut, Beijing 100871, Peoples R China
[3] Peking Univ, Shenzhen Grad Sch, Lab Chem Genom, Beijing 100871, Peoples R China
来源：
JOURNAL OF COMBINATORIAL CHEMISTRY | 2005年 / 7卷 / 06期
关键词：
D O I：
10.1021/cc050099b
中图分类号：
O69 [应用化学];
学科分类号：
081704 ;
摘要：
A one-pot synthesis of diverse benzofurans and indoles from readily available starting materials was achieved via the sequential Ugi four-component reaction, intramolecular Diels-Alder reaction, and oxidative aromatization.
引用
收藏
页码：958 / 967
页数：10
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