Stable σ-adducts of 5-azauracil with C-nucleophiles

被引:0
作者
Azev, YA [1 ]
Shorshnev, SV
Gabel, D
机构
[1] Urals Sci Res Int Technol Med Preparat, Ekaterinburg 620219, Russia
[2] ChemBridge, Moscow 119435, Russia
[3] Univ Bremen, Dept Chem, D-28334 Bremen, Germany
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
The heating of 5-azauracil 1 with malonamide in butanol resulted in 1,2,3,4,5,6-hexahydro-6-(dicarbamoylmethyl)-1,3,5-triazine-2,4-dione 3. Under conditions of acid catalysis, compound I reacted with o-phenylenediamine, pyrrogallol, resorcinol and phenylhydrazine derivatives to form the corresponding 6-derivatives of 1,2,3,4,5,6-hexahydro- 1,3,5-triazine-2,4-dione.
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页码:234 / 235
页数:2
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