ONE-POT SYNTHESIS OF HYDROXYBENZO[d]OXAZOLE-2-ALIPHATIC ACID DERIVATIVES BY MEERWEIN'S REAGENT

被引：2

作者：

Zhang, Wei ^{[1
]}

Liu, Wenlu ^{[1
]}

Jiang, Xizhen ^{[1
]}

Jiang, Faqin ^{[1
]}

Fu, Lei ^{[1
]}

机构：

[1] Shanghai Jiao Tong Univ, Sch Pharm, Shanghai 200240, Peoples R China

来源：

SYNTHETIC COMMUNICATIONS | 2012年 / 42卷 / 18期

关键词：

2-Aminophenol; benzo[d]oxazole; Meerwein's reagent; triethyloxonium tetrafluoroborate; BENZOXAZOLE DERIVATIVES; INHIBITORS; BENZIMIDAZOLES; ANALOGS;

D O I：

10.1080/00397911.2011.567435

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A general one-pot synthesis of hydroxylbenzo[d]oxazole-2-aliphatic acid esters and hydroxylbenzo[d]oxazole-2-amino acid esters was successfully achieved in good yield by using Meerwein's reagent.

引用

页码：2772 / 2779

页数：8

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