共 11 条
Specific Aldosterone Synthase Inhibition: A Potential Improvement Over Mineralocorticoid Receptor Antagonism?
被引:0
作者:

Schneider, Markus P.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Erlangen Nurnberg, Dept Hypertens & Nephrol, Erlangen, Germany Univ Erlangen Nurnberg, Dept Hypertens & Nephrol, Erlangen, Germany

Hilgers, Karl F.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Erlangen Nurnberg, Dept Hypertens & Nephrol, Erlangen, Germany Univ Erlangen Nurnberg, Dept Hypertens & Nephrol, Erlangen, Germany
机构:
[1] Univ Erlangen Nurnberg, Dept Hypertens & Nephrol, Erlangen, Germany
关键词:
DOUBLE-BLIND;
HYPERTENSION;
DEOXYCORTICOSTERONE;
PLACEBO;
DISEASE;
TRIAL;
D O I:
10.1161/HYPERTENSIONAHA.116.07939
中图分类号:
R6 [外科学];
学科分类号:
1002 ;
100210 ;
摘要:
引用
收藏
页码:11 / 12
页数:2
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共 11 条
- [1] Aldosterone Synthase Inhibition With LCI699 A Proof-of-Concept Study in Patients With Primary Aldosteronism[J]. HYPERTENSION, 2010, 56 (05) : 831 - +论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Peyrard, Severine论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 05, Fac Med, Paris, France Hop Europeen Georges Pompidou, APHP, INSERM, Clin Invest Ctr 9201, F-75015 Paris, FranceWatson, Catherine论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Hop Europeen Georges Pompidou, APHP, INSERM, Clin Invest Ctr 9201, F-75015 Paris, FrancePlouin, Pierre-Francois论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 05, Fac Med, Paris, France Hop Europeen Georges Pompidou, APHP, INSERM, Clin Invest Ctr 9201, F-75015 Paris, France
- [2] Preclinical and Early Clinical Profile of a Highly Selective and Potent Oral Inhibitor of Aldosterone Synthase (CYP11B2)[J]. HYPERTENSION, 2017, 69 (01) : 189 - 196Bogman, Katrijn论文数: 0 引用数: 0 h-index: 0机构: Roche Innovat Ctr Basel, Pharma Res & Early Dev, Clin Pharmacol, Basel, Switzerland Roche Innovat Ctr Basel, Pharma Res & Early Dev, Clin Pharmacol, Basel, SwitzerlandSchwab, Dietmar论文数: 0 引用数: 0 h-index: 0机构: Roche Innovat Ctr Basel, Pharma Res & Early Dev, Clin Pharmacol, Basel, Switzerland Roche Innovat Ctr Basel, Pharma Res & Early Dev, Clin Pharmacol, Basel, SwitzerlandDelporte, Marie-Laure论文数: 0 引用数: 0 h-index: 0机构: Roche Innovat Ctr Basel, Pharma Res & Early Dev, Clin Pharmacol, Basel, Switzerland Roche Innovat Ctr Basel, Pharma Res & Early Dev, Clin Pharmacol, Basel, SwitzerlandPalermo, Giuseppe论文数: 0 引用数: 0 h-index: 0机构: Roche Innovat Ctr Basel, Pharma Res & Early Dev, Biostat, Basel, Switzerland Roche Innovat Ctr Basel, Pharma Res & Early Dev, Clin Pharmacol, Basel, SwitzerlandAmrein, Kurt论文数: 0 引用数: 0 h-index: 0机构: Roche Innovat Ctr Basel, Pharma Res & Early Dev, Discovery, Basel, Switzerland Roche Innovat Ctr Basel, Pharma Res & Early Dev, Clin Pharmacol, Basel, SwitzerlandMohr, Susanne论文数: 0 引用数: 0 h-index: 0机构: Roche Innovat Ctr Basel, Pharma Res & Early Dev, Pharmaceut Sci, Basel, Switzerland Roche Innovat Ctr Basel, Pharma Res & Early Dev, Clin Pharmacol, Basel, SwitzerlandMudry, Maria Cristina De Vera论文数: 0 引用数: 0 h-index: 0机构: Roche Innovat Ctr Basel, Pharma Res & Early Dev, Pharmaceut Sci, Basel, Switzerland Roche Innovat Ctr Basel, Pharma Res & Early Dev, Clin Pharmacol, Basel, SwitzerlandBrown, Morris J.论文数: 0 引用数: 0 h-index: 0机构: Queen Mary Univ London, William Harvey Res Inst, Clin Pharmacol, London, England Roche Innovat Ctr Basel, Pharma Res & Early Dev, Clin Pharmacol, Basel, SwitzerlandFerber, Philippe论文数: 0 引用数: 0 h-index: 0机构: Roche Innovat Ctr Basel, Pharma Res & Early Dev, Translat Med, Cardiovasc Dis, Basel, Switzerland Roche Innovat Ctr Basel, Pharma Res & Early Dev, Clin Pharmacol, Basel, Switzerland
- [3] Effects of a Novel Aldosterone Synthase Inhibitor for Treatment of Primary Hypertension Results of a Randomized, Double-Blind, Placebo- and Active-Controlled Phase 2 Trial[J]. CIRCULATION, 2011, 124 (18) : 1945 - U124Calhoun, David A.论文数: 0 引用数: 0 h-index: 0机构: Univ Alabama, Vasc Biol & Hypertens Program, Birmingham, AL 35294 USA Univ Alabama, Vasc Biol & Hypertens Program, Birmingham, AL 35294 USAWhite, William B.论文数: 0 引用数: 0 h-index: 0机构: Univ Connecticut, Sch Med, Div Hypertens & Clin Pharmacol, Pat & Jim Calhoun Cardiol Ctr, Farmington, CT USA Univ Alabama, Vasc Biol & Hypertens Program, Birmingham, AL 35294 USAKrum, Henry论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Ctr Cardiovasc Res & Educ Therapeut, Dept Epidemiol & Prevent Med, Melbourne, Vic 3004, Australia Univ Alabama, Vasc Biol & Hypertens Program, Birmingham, AL 35294 USAGuo, Weinong论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Alabama, Vasc Biol & Hypertens Program, Birmingham, AL 35294 USABermann, Georgina论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Basel, Switzerland Univ Alabama, Vasc Biol & Hypertens Program, Birmingham, AL 35294 USATrapani, Angelo论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Alabama, Vasc Biol & Hypertens Program, Birmingham, AL 35294 USALefkowitz, Martin P.论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Alabama, Vasc Biol & Hypertens Program, Birmingham, AL 35294 USAMenard, Joel论文数: 0 引用数: 0 h-index: 0机构: INSERM, CIC 9201, Paris, France Univ Paris 05, Paris, France Univ Alabama, Vasc Biol & Hypertens Program, Birmingham, AL 35294 USA
- [4] Mineralocorticoid Receptors, Salt-Sensitive Hypertension, and Metabolic Syndrome[J]. HYPERTENSION, 2010, 55 (04) : 813 - 818Fujita, Toshiro论文数: 0 引用数: 0 h-index: 0机构: Univ Tokyo, Dept Nephrol & Endocrinol, Sch Med, Bunkyo Ku, Tokyo 1138655, Japan Univ Tokyo, Dept Nephrol & Endocrinol, Sch Med, Bunkyo Ku, Tokyo 1138655, Japan
- [5] The role of aldosterone and mineralocorticoid receptors in cardiovascular disease[J]. AMERICAN JOURNAL OF CARDIOVASCULAR DRUGS, 2007, 7 (03) : 151 - 157Funder, John W.论文数: 0 引用数: 0 h-index: 0机构: Prince Henrys Inst Med Res, Clayton, Vic 3168, Australia Prince Henrys Inst Med Res, Clayton, Vic 3168, Australia
- [6] Spironolactone Reduces Cardiovascular and Cerebrovascular Morbidity and Mortality in Hemodialysis Patients[J]. JOURNAL OF THE AMERICAN COLLEGE OF CARDIOLOGY, 2014, 63 (06) : 529 - 536Matsumoto, Yoshihiro论文数: 0 引用数: 0 h-index: 0机构: Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, Japan Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, JapanMori, Yasuo论文数: 0 引用数: 0 h-index: 0机构: Shibukawa Clin, Shizuoka, Japan Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, JapanKageyama, Shinji论文数: 0 引用数: 0 h-index: 0机构: Kageyama Urol Clin, Shizuoka, Japan Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, JapanArihara, Kazuo论文数: 0 引用数: 0 h-index: 0机构: Ohtemachi Clin, Shizuoka, Japan Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, JapanSugiyama, Toshikazu论文数: 0 引用数: 0 h-index: 0机构: Sugiyama Clin, Shizuoka, Japan Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, JapanOhmura, Hiromichi论文数: 0 引用数: 0 h-index: 0机构: Sugawara Clin, Shizuoka, Japan Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, JapanYakushigawa, Toru论文数: 0 引用数: 0 h-index: 0机构: Shibukawa Clin, Shizuoka, Japan Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, JapanSugiyama, Hatsumi论文数: 0 引用数: 0 h-index: 0机构: Sugiyama Clin, Shizuoka, Japan Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, JapanShimada, Yasushi论文数: 0 引用数: 0 h-index: 0机构: Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, Japan Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, JapanNojima, Youichi论文数: 0 引用数: 0 h-index: 0机构: Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, Japan Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, JapanShio, Nobuo论文数: 0 引用数: 0 h-index: 0机构: Kageyama Urol Clin, Shizuoka, Japan Shizuoka City Hospital, Dept Nephrol & Dialysis, Aoi Ku, Shizuoka 4208630, Japan
- [7] Aldosterone synthase inhibition: cardiorenal protection in animal disease models and translation of hormonal effects to human subjects[J]. JOURNAL OF TRANSLATIONAL MEDICINE, 2014, 12Menard, Joel论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 05, Fac Med, Paris, France Georges Pompidou Hosp, AP HP, INSERM, Clin Invest Ctr, Paris, France Univ Paris 05, Fac Med, Paris, FranceRigel, Dean F.论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Paris 05, Fac Med, Paris, FranceWatson, Catherine论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Cambridge, MA 02139 USA Univ Paris 05, Fac Med, Paris, FranceJeng, Arco Y.论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Paris 05, Fac Med, Paris, FranceFu, Fumin论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Paris 05, Fac Med, Paris, FranceBeil, Michael论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Paris 05, Fac Med, Paris, FranceLiu, Jing论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Paris 05, Fac Med, Paris, FranceChen, Wei论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Paris 05, Fac Med, Paris, FranceHu, Chii-Whei论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Paris 05, Fac Med, Paris, FranceLeung-Chu, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Paris 05, Fac Med, Paris, FranceLaSala, Daniel论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Paris 05, Fac Med, Paris, FranceLiang, Guiqing论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Cambridge, MA 02139 USA Univ Paris 05, Fac Med, Paris, FranceRebello, Sam论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Paris 05, Fac Med, Paris, FranceZhang, Yiming论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, E Hanover, NJ USA Univ Paris 05, Fac Med, Paris, FranceDole, William P.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Cambridge, MA 02139 USA Univ Paris 05, Fac Med, Paris, France
- [8] Deoxycorticosterone inactivation by AKR1C3 in human mineralocorticoid target tissues[J]. MOLECULAR AND CELLULAR ENDOCRINOLOGY, 2006, 248 (1-2) : 79 - 86Sharma, KK论文数: 0 引用数: 0 h-index: 0机构: Univ Texas, SW Med Ctr, Dept Obstet Gynecol & Biochem, Dallas, TX 75230 USALindqvist, A论文数: 0 引用数: 0 h-index: 0机构: Univ Texas, SW Med Ctr, Dept Obstet Gynecol & Biochem, Dallas, TX 75230 USAZhou, XJ论文数: 0 引用数: 0 h-index: 0机构: Univ Texas, SW Med Ctr, Dept Obstet Gynecol & Biochem, Dallas, TX 75230 USAAuchus, RJ论文数: 0 引用数: 0 h-index: 0机构: Univ Texas, SW Med Ctr, Dept Obstet Gynecol & Biochem, Dallas, TX 75230 USAPenning, TM论文数: 0 引用数: 0 h-index: 0机构: Univ Texas, SW Med Ctr, Dept Obstet Gynecol & Biochem, Dallas, TX 75230 USAAndersson, S论文数: 0 引用数: 0 h-index: 0机构: Univ Texas, SW Med Ctr, Dept Obstet Gynecol & Biochem, Dallas, TX 75230 USA Univ Texas, SW Med Ctr, Dept Obstet Gynecol & Biochem, Dallas, TX 75230 USA
- [9] The mislabelling of deoxycorticosterone: making sense of corticosteroid structure and function[J]. JOURNAL OF ENDOCRINOLOGY, 2011, 211 (01) : 3 - 16Vinson, Gavin P.论文数: 0 引用数: 0 h-index: 0机构: Queen Mary Univ London, Sch Biol & Chem Sci, London E1 4NS, England Queen Mary Univ London, Sch Biol & Chem Sci, London E1 4NS, England
- [10] 24 HOUR PATTERN OF EPISODIC SECRETION OF CORTISOL IN NORMAL SUBJECTS[J]. JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1971, 33 (01) : 14 - +WEITZMAN, ED论文数: 0 引用数: 0 h-index: 0FUKUSHIMA, D论文数: 0 引用数: 0 h-index: 0NOGEIRE, C论文数: 0 引用数: 0 h-index: 0ROFFWARG, H论文数: 0 引用数: 0 h-index: 0GALLAGHER, TF论文数: 0 引用数: 0 h-index: 0HELLMAN, L论文数: 0 引用数: 0 h-index: 0