共 33 条
[1]
[Anonymous], 2000, Eurofins (Millipore), Patent No. [WO 2007070398, 2007070398]
[2]
Flipped out: Structure-guided design of selective pyrazolylpyrrole ERK inhibitors
[J].
Aronov, Alex M.
;
Baker, Christopher
;
Bemis, Guy W.
;
Cao, Jingrong
;
Chen, Guanjing
;
Ford, Pamella J.
;
Germann, Ursula A.
;
Green, Jeremy
;
Hale, Michael R.
;
Jacobs, Marc
;
Janetka, James W.
;
Maltais, Francois
;
Martinez-Botella, Gabriel
;
Namchuk, Mark N.
;
Straub, Judy
;
Tang, Qing
;
Xie, Xiaoling
.
JOURNAL OF MEDICINAL CHEMISTRY,
2007, 50 (06)
:1280-1287

Aronov, Alex M.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Baker, Christopher
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Bemis, Guy W.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Cao, Jingrong
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Chen, Guanjing
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Ford, Pamella J.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Germann, Ursula A.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Green, Jeremy
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Hale, Michael R.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Jacobs, Marc
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Janetka, James W.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Maltais, Francois
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Martinez-Botella, Gabriel
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Namchuk, Mark N.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Straub, Judy
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Tang, Qing
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Xie, Xiaoling
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA
[3]
Structure-Guided Design of Potent and Selective Pyrimidylpyrrole Inhibitors of Extracellular Signal-Regulated Kinase (ERK) Using Conformational Control
[J].
Aronov, Alex M.
;
Tang, Qing
;
Martinez-Botella, Gabriel
;
Bemis, Guy W.
;
Cao, Jingrong
;
Chen, Guanjing
;
Ewing, Nigel P.
;
Ford, Pamella J.
;
Germann, Ursula A.
;
Green, Jeremy
;
Hale, Michael R.
;
Jacobs, Marc
;
Janetka, James W.
;
Maltais, Francois
;
Markland, William
;
Namchuk, Mark N.
;
Nanthakumar, Suganthini
;
Poondru, Srinivasu
;
Straub, Judy
;
ter Haar, Ernst
;
Xie, Xiaoling
.
JOURNAL OF MEDICINAL CHEMISTRY,
2009, 52 (20)
:6362-6368

Aronov, Alex M.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Tang, Qing
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Martinez-Botella, Gabriel
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Bemis, Guy W.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Cao, Jingrong
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Chen, Guanjing
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Ewing, Nigel P.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Ford, Pamella J.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Germann, Ursula A.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Green, Jeremy
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Hale, Michael R.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Jacobs, Marc
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Janetka, James W.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Maltais, Francois
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Markland, William
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Namchuk, Mark N.
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Nanthakumar, Suganthini
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Poondru, Srinivasu
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Straub, Judy
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

ter Haar, Ernst
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA

Xie, Xiaoling
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut Inc, Cambridge, MA 02139 USA Vertex Pharmaceut Inc, Cambridge, MA 02139 USA
[4]
Barlaam B. C., 2009, Patent, Patent No. [WO 2009153589, 2012036997, WO 2012036997]
[5]
Barlaam B.C., 2009, Patent, Patent No. [WO 2009153589, 2009153589, WO2009/153589]
[6]
Discovery of 5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine inhibitors of Erk2
[J].
Blake, James F.
;
Gaudino, John J.
;
De Meese, Jason
;
Mohr, Peter
;
Chicarelli, Mark
;
Tian, Hongqi
;
Garrey, Rustam
;
Thomas, Allen
;
Siedem, Christopher S.
;
Welch, Michael B.
;
Kolakowski, Gabrielle
;
Kaus, Robert
;
Burkard, Michael
;
Martinson, Matthew
;
Chen, Huifen
;
Dean, Brian
;
Dudley, Danette A.
;
Gould, Stephen E.
;
Pacheco, Patricia
;
Shahidi-Latham, Sheerin
;
Wang, Weiru
;
West, Kristina
;
Yin, Jianping
;
Moffat, John
;
Schwarz, Jacob B.
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
2014, 24 (12)
:2635-2639

Blake, James F.
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Gaudino, John J.
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

De Meese, Jason
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Mohr, Peter
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Chicarelli, Mark
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Tian, Hongqi
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Garrey, Rustam
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Thomas, Allen
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Siedem, Christopher S.
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Welch, Michael B.
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Kolakowski, Gabrielle
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Kaus, Robert
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Burkard, Michael
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Martinson, Matthew
论文数: 0 引用数: 0
h-index: 0
机构:
Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USA

Chen, Huifen
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA

Dean, Brian
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA

Dudley, Danette A.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA

Gould, Stephen E.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA

Pacheco, Patricia
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA

Shahidi-Latham, Sheerin
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA

Wang, Weiru
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA

West, Kristina
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA

Yin, Jianping
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA

Moffat, John
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA

Schwarz, Jacob B.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA
[7]
Discovery of Novel, Dual Mechanism ERK Inhibitors by Affinity Selection Screening of an Inactive Kinase
[J].
Deng, Yongqi
;
Shipps, Gerald W., Jr.
;
Cooper, Alan
;
English, Jessie M.
;
Annis, D. Allen
;
Carr, Donna
;
Nan, Yang
;
Wang, Tong
;
Zhu, Hugh Y.
;
Chuang, Cheng-Chi
;
Dayananth, Priya
;
Hruza, Alan W.
;
Xiao, Li
;
Jin, Weihong
;
Kirschmeier, Paul
;
Windsor, William T.
;
Samatar, Ahmed A.
.
JOURNAL OF MEDICINAL CHEMISTRY,
2014, 57 (21)
:8817-8826

Deng, Yongqi
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USA

Shipps, Gerald W., Jr.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USA

Cooper, Alan
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Boston, MA 02115 USA

English, Jessie M.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Boston, MA 02115 USA

Annis, D. Allen
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USA

Carr, Donna
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Boston, MA 02115 USA

Nan, Yang
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USA

Wang, Tong
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USA

Zhu, Hugh Y.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Boston, MA 02115 USA

Chuang, Cheng-Chi
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USA

Dayananth, Priya
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Boston, MA 02115 USA

Hruza, Alan W.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Boston, MA 02115 USA

Xiao, Li
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Boston, MA 02115 USA

Jin, Weihong
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Boston, MA 02115 USA

Kirschmeier, Paul
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Boston, MA 02115 USA

Windsor, William T.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Boston, MA 02115 USA

Samatar, Ahmed A.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Boston, MA 02115 USA
[8]
MAP kinase signalling pathways in cancer
[J].
Dhillon, A. S.
;
Hagan, S.
;
Rath, O.
;
Kolch, W.
.
ONCOGENE,
2007, 26 (22)
:3279-3290

Dhillon, A. S.
论文数: 0 引用数: 0
h-index: 0
机构: Beatson Inst Canc Res, Glasgow G61 1BD, Lanark, Scotland

Hagan, S.
论文数: 0 引用数: 0
h-index: 0
机构: Beatson Inst Canc Res, Glasgow G61 1BD, Lanark, Scotland

Rath, O.
论文数: 0 引用数: 0
h-index: 0
机构: Beatson Inst Canc Res, Glasgow G61 1BD, Lanark, Scotland

论文数: 引用数:
h-index:
机构:
[9]
MEK1 mutations confer resistance to MEK and B-RAF inhibition
[J].
Emery, Caroline M.
;
Vijayendran, Krishna G.
;
Zipser, Marie C.
;
Sawyer, Allison M.
;
Niu, Lili
;
Kim, Jessica J.
;
Hatton, Charles
;
Chopra, Rajiv
;
Oberholzer, Patrick A.
;
Karpova, Maria B.
;
MacConaill, Laura E.
;
Zhang, Jianming
;
Gray, Nathanael S.
;
Sellers, William R.
;
Dummer, Reinhard
;
Garraway, Levi A.
.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
2009, 106 (48)
:20411-20416

Emery, Caroline M.
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA
Harvard Univ, Sch Med, Dana Farber Canc Inst, Ctr Canc Genome Discovery, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Vijayendran, Krishna G.
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA
Harvard Univ, Sch Med, Dana Farber Canc Inst, Ctr Canc Genome Discovery, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Zipser, Marie C.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Zurich Hosp, Dept Dermatol, CH-8091 Zurich, Switzerland Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Sawyer, Allison M.
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA
Harvard Univ, Sch Med, Dana Farber Canc Inst, Ctr Canc Genome Discovery, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Niu, Lili
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA
Harvard Univ, Sch Med, Dana Farber Canc Inst, Ctr Canc Genome Discovery, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Kim, Jessica J.
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA
Harvard Univ, Sch Med, Dana Farber Canc Inst, Ctr Canc Genome Discovery, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Hatton, Charles
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA
Harvard Univ, Sch Med, Dana Farber Canc Inst, Ctr Canc Genome Discovery, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Chopra, Rajiv
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst BioMed Res, Cambridge, MA 02139 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Oberholzer, Patrick A.
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA
Harvard Univ, Sch Med, Dana Farber Canc Inst, Ctr Canc Genome Discovery, Boston, MA 02115 USA
Univ Zurich Hosp, Dept Dermatol, CH-8091 Zurich, Switzerland
Broad Inst, Cambridge, MA 02142 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Karpova, Maria B.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Zurich Hosp, Dept Dermatol, CH-8091 Zurich, Switzerland Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

MacConaill, Laura E.
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA
Harvard Univ, Sch Med, Dana Farber Canc Inst, Ctr Canc Genome Discovery, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Zhang, Jianming
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Gray, Nathanael S.
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Sellers, William R.
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst BioMed Res, Cambridge, MA 02139 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Dummer, Reinhard
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Zurich Hosp, Dept Dermatol, CH-8091 Zurich, Switzerland Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA

Garraway, Levi A.
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA
Harvard Univ, Sch Med, Dana Farber Canc Inst, Ctr Canc Genome Discovery, Boston, MA 02115 USA
Broad Inst, Cambridge, MA 02142 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA
[10]
Discovery of a Potent and Selective EGFR Inhibitor (AZD9291) of Both Sensitizing and T790M Resistance Mutations That Spares the Wild Type Form of the Receptor
[J].
Finlay, M. Raymond V.
;
Anderton, Mark
;
Ashton, Susan
;
Ballard, Peter
;
Bethel, Paul A.
;
Box, Matthew R.
;
Bradbury, Robert H.
;
Brown, Simon J.
;
Butterworth, Sam
;
Campbell, Andrew
;
Chorley, Christopher
;
Colclough, Nicola
;
Cross, Darren A. E.
;
Currie, Gordon S.
;
Grist, Matthew
;
Hassall, Lorraine
;
Hill, George B.
;
James, Daniel
;
James, Michael
;
Kemmitt, Paul
;
Klinowska, Teresa
;
Lamont, Gillian
;
Lamont, Scott G.
;
Martin, Nathaniel
;
McFarland, Heather L.
;
Mellor, Martine J.
;
Orme, Jonathon P.
;
Perkins, David
;
Perkins, Paula
;
Richmond, Graham
;
Smith, Peter
;
Ward, Richard A.
;
Waring, Michael J.
;
Whittaker, David
;
Wells, Stuart
;
Wrigley, Gail L.
.
JOURNAL OF MEDICINAL CHEMISTRY,
2014, 57 (20)
:8249-8267

Finlay, M. Raymond V.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Anderton, Mark
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Drug Safety & Metab, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Ashton, Susan
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Ballard, Peter
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Bethel, Paul A.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Box, Matthew R.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Bradbury, Robert H.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Brown, Simon J.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Butterworth, Sam
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Campbell, Andrew
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Chorley, Christopher
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Colclough, Nicola
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Drug Safety & Metab, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Cross, Darren A. E.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Currie, Gordon S.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Grist, Matthew
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Hassall, Lorraine
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Hill, George B.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

James, Daniel
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

James, Michael
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Kemmitt, Paul
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Klinowska, Teresa
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Lamont, Gillian
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Lamont, Scott G.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Martin, Nathaniel
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

McFarland, Heather L.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Global Med Dev, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Mellor, Martine J.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Orme, Jonathon P.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Perkins, David
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Perkins, Paula
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Richmond, Graham
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Smith, Peter
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Ward, Richard A.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Waring, Michael J.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Whittaker, David
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Wells, Stuart
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England

Wrigley, Gail L.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Oncol Innovat Med, Macclesfield SK10 4TG, Cheshire, England