A novel multi-component synthesis of 4-arylaminoquinazolines

被引:46
作者
Heravi, Majid M. [1 ]
Sadjadi, Samaheh [1 ]
Haj, Negar Mokhtari [1 ]
Oskooie, Hossein A. [1 ]
Shoar, Rahim Hekmat [1 ]
Bamoharram, Fatemeh F. [2 ]
机构
[1] Alzahra Univ, Sch Sci, Dept Chem, Tehran, Iran
[2] Islamic Azad Univ, Mashhad Branch, Dept Chem, Mashhad, Iran
关键词
4-Arylaminoquinazoline; Recyclable catalyst; Heteropolyacid; Keggin; GROWTH-FACTOR RECEPTOR; RECYCLABLE CATALYSTS; TYROSINE KINASE; HETEROPOLYACIDS; QUINAZOLIN-4(3H)-ONES; QUINAZOLINES; INHIBITORS; MICROWAVE; GREEN; SITE;
D O I
10.1016/j.tetlet.2008.12.044
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A new multi-component synthesis of 4-arylaminoquinazolines from the reaction of 2-aminobenzamide, orthoesters, and substituted anilines in the presence of catalytic amounts of Keggin-type heteropolyacids is reported. The effects of reaction conditions and different heteropolyacids have been studied. (C) 2008 Elsevier Ltd. All rights reserved.
引用
收藏
页码:943 / 945
页数:3
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