4-Alkyl-6-amino-N 3,N 5-diaryl-2-thioxo-1,2,3,4-tetrahydropyridine-3,5-dicarboxamides: II. Synthesis and selected reactions

被引：4

作者：

Dyachenko, V. D. ^{[1
]}

Karpov, E. N. ^{[1
]}

Feskov, I. A. ^{[1
]}

机构：

[1] Taras Shevchenko Luhansk Natl Univ, UA-91011 Lugansk, Ukraine

来源：

RUSSIAN JOURNAL OF GENERAL CHEMISTRY | 2013年 / 83卷 / 09期

关键词：

ALIPHATIC-ALDEHYDES; 4H-PYRANS;

D O I：

10.1134/S1070363213090156

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

New 4-alkyl-6-amino-N (3),N (5)-diaryl-2-thioxo-1,2,3,4-tetrahydropyridine-3,5-dicarboxamides have been prepared via enantioselective reaction of 3-amino-N-aryl-3-thioxopropanamides with N-aryl-2-cyanoacetamide and aliphatic aldehydes. The prepared products can be regioselectively alkylated at sulfur atom.

引用

页码：1716 / 1723

页数：8

共 30 条

[1]

[Anonymous], 2000, Structure Determination of organic compounds

[2]

Barton D., 1979, COMPREHENSIVE ORGANI, V1st

[3]

Brytsun V.N., 2012, 2 FUNKTSIOINALIZIROV

[4]

Deyanov A.B., 2004, CHEM HETEROCYCL COMP, V12, P1560

[5]

Dyachenko A.D., 2004, CHEM HETEROCYCL COMP, P1009

[6]

Dyachenko A.D., 2003, CHEM HETEROCYCL COMP, P744

[7]

Dyachenko A.D., 2004, CHEM HETEROCYCL COMP, P650

[8] SYNTHESIS AND ALKYLATION OF N(3)-ARYL-N(5)-PHENYL-6-AMINO-4-ARYL(2-FURYL)-2-THIOXO-1,2,3,4-TETRAHYDROPYRIDINE-3,5-DICARBOXAMIDE [J].

Dyachenko, V. D. ;

Krasnikov, D. A. ;

Khorik, M. V. .

CHEMISTRY OF HETEROCYCLIC COMPOUNDS, 2008, 44 (07) :815-819

[9] Aliphatic aldehydes in multicomponent syntheses of 4-alkyl-substituted partially hydrogenated quinolines, fused 4H-pyrans, and 2-amino-4-ethyl-5-methylbenzene-1,3-dicarbonitrile [J].

Dyachenko, V. D. ;

Chernega, A. N. .

RUSSIAN JOURNAL OF ORGANIC CHEMISTRY, 2006, 42 (04) :567-576

[10] 4-alkyl-6-amino-4-N3,N5-diaryl-2-thioxo-1,2,3,4-tetrahydropyridine-3,5-dicarboxamides: I. Tandem synthesis and alkylation. Molecular and crystal structure of 6-allylsulfanyl-2-amino-4-isobutyl-N3,N5-di-m-tolyl-3,4-dihydropyridine-3,5-dicarboxamide [J].

Dyachenko, V. D. ;

Karpov, E. N. .

RUSSIAN JOURNAL OF GENERAL CHEMISTRY, 2013, 83 (07) :1394-1401

← 1 2 3 →