Reactivity as glycine templates of 1,2-dialkyl-2,4-dihydro-1H-pyrazino[2,1-b]quinazoline-3,6-diones

被引：13
作者：
Buenadicha, FL [1 ]
Avendaño, C [1 ]
Söllhuber, M [1 ]
机构：
[1] Univ Complutense, Dept Quim Organ & Farmaceut, E-28040 Madrid, Spain
来源：
TETRAHEDRON-ASYMMETRY | 2001年 / 12卷 / 21期
关键词：
D O I：
10.1016/S0957-4166(01)00515-8
中图分类号：
O61 [无机化学];
学科分类号：
070301 ; 081704 ;
摘要：
The 1-methyl(iso-propyl)-2-benzyl-2,4-dihydro-1H-pyrazino[2,1-b]quinazoline-3,6-diones 8 and 9 could be regio- and diastereoselectively alkylated at C(4) with retention of configuration at both stereocentres. (C) 2002 Elsevier Science Ltd. All rights reserved.
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收藏
页码：3019 / 3028
页数：10
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