The reactions of diacetylenic ketones with nitrogen nucleophiles; facile preparation of alkynyl substituted pyrimidines and pyrazoles

被引:45
作者
Baldwin, JE
Pritchard, GJ
Rathmell, RE
机构
[1] Univ Oxford, Dyson Perrins Lab, Oxford OX1 3QY, England
[2] Univ Loughborough, Dept Chem, Loughborough LE11 3TU, Leics, England
来源
JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 2001年 / 22期
关键词
D O I
10.1039/b108645f
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Alkynyl substituted pyrimidines and pyrazoles have been synthesized by cyclocondensations of diacetylenic ketones with amidines and hydrazines.
引用
收藏
页码:2906 / 2908
页数:3
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