Synthesis and evaluation of new triazolobenzothiazole derivatives as potential anti-tubercular agents

被引：0

作者：

Paranjape, SD ^{[1
]}

Bobade, AS ^{[1
]}

Khadse, BG ^{[1
]}

机构：

[1] Haffkine Inst, Dept Chemotherapy, Bombay 400012, Maharashtra, India

来源：

ARZNEIMITTEL-FORSCHUNG-DRUG RESEARCH | 2001年 / 51卷 / 11期

关键词：

Mycobacterium tuberculosis; sulfonamides; triazolobenzothiazoles; antitubercular activity; S-benzyl derivatives;

D O I：

暂无

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

A series of sulfonamides and S-benzyl derivatives of substituted/unsubstituted S-triazolo-(3,4,-b)-benzothiazole-3-thiones were synthesized. These triazolobenzothiazole derivatives were evaluated for antitubercular activity against H(37)Rv strain of Mycobacterium tuberculosis. A number of promising compounds have been obtained.

引用

页码：916 / 919

页数：4

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