共 8 条
- [1] Discovery of YAP-TEAD protein-protein interaction (PPI) inhibitors for cancer therapyCANCER RESEARCH, 2016, 76Soude, Anne论文数: 0 引用数: 0 h-index: 0Barth, Martine论文数: 0 引用数: 0 h-index: 0Bocart, Stephanie论文数: 0 引用数: 0 h-index: 0Thoreau, Frederic论文数: 0 引用数: 0 h-index: 0Masson, Philippe论文数: 0 引用数: 0 h-index: 0Braccini, Isabelle论文数: 0 引用数: 0 h-index: 0Montalbetti, Christian论文数: 0 引用数: 0 h-index: 0Brogue, Pierre论文数: 0 引用数: 0 h-index: 0Fromond, Claudia论文数: 0 引用数: 0 h-index: 0
- [2] Discovery of YAP-TEAD protein-protein interaction inhibitors (PPI) for treating malignant pleural mesothelioma (MPM).MOLECULAR CANCER RESEARCH, 2020, 18 (08) : 49 - 49Soude, Anne论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceBarth, Martine论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceLuccarini, Jean-Michel论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceDelaporte, Severine论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceChirade, Florence论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceValaire, Christelle论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceBoulay, Aude论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceCheret, Genevieve论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceDorchie, Marie论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceEstivalet, Celine论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceTuya-Boustugue, Pascale论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceTranchand, Robin论文数: 0 引用数: 0 h-index: 0机构: INSERM, URMS 1138, Paris, France Inventiva, Daix, FranceJean, Didier论文数: 0 引用数: 0 h-index: 0机构: INSERM, URMS 1138, Paris, France Inventiva, Daix, FranceQuetel, Lisa论文数: 0 引用数: 0 h-index: 0机构: INSERM, URMS 1138, Paris, France Inventiva, Daix, FranceAssie, Jean-Baptiste论文数: 0 引用数: 0 h-index: 0机构: INSERM, URMS 1138, Paris, France Inventiva, Daix, FranceKonstantinova, Irena论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceJunien, Jean-Louis论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceBroqua, Pierre论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, France
- [3] A novel anti-cancer compound development targeting YAP-TEAD protein-protein interactionEUROPEAN JOURNAL OF CANCER, 2022, 174 : S37 - S37Park, J. S.论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South KoreaShin, Y. K.论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ, Gangnam Severance Biomed Res Ctr, Coll Med, Seoul, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South KoreaHong, E.论文数: 0 引用数: 0 h-index: 0机构: Daegu Gyeongbuk Med Innovat Fdn, New Drug Dev Ctr, Daegu, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South KoreaPark, Y. H.论文数: 0 引用数: 0 h-index: 0机构: Daegu Gyeongbuk Med Innovat Fdn, New Drug Dev Ctr, Daegu, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South KoreaUm, J.论文数: 0 引用数: 0 h-index: 0机构: Samjin Pharmaceut Co Ltd, Res Ctr, Seoul, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South KoreaLee, D.论文数: 0 引用数: 0 h-index: 0机构: Samjin Pharmaceut Co Ltd, Res Ctr, Seoul, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South KoreaKwon, H. S.论文数: 0 引用数: 0 h-index: 0机构: Samjin Pharmaceut Co Ltd, Res Ctr, Seoul, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South KoreaIssabayeva, G.论文数: 0 引用数: 0 h-index: 0机构: Korea Res Inst Chem Technol, Therapeut Biotechnol Div Dept Drug Discovery, Daejeon, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South KoreaKang, O. Y.论文数: 0 引用数: 0 h-index: 0机构: Korea Res Inst Chem Technol, Therapeut Biotechnol Div Dept Drug Discovery, Daejeon, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South KoreaLim, B. H.论文数: 0 引用数: 0 h-index: 0机构: Korea Res Inst Chem Technol, Therapeut Biotechnol Div Dept Drug Discovery, Daejeon, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South KoreaPark, S. J.论文数: 0 引用数: 0 h-index: 0机构: Korea Res Inst Chem Technol, Therapeut Biotechnol Div Dept Drug Discovery, Daejeon, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South KoreaLim, H. J.论文数: 0 引用数: 0 h-index: 0机构: Korea Res Inst Chem Technol, Therapeut Biotechnol Div Dept Drug Discovery, Daejeon, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South KoreaJeung, H. C.论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ, Div Med Oncol Dept Internal Med, Gangnam Severance Hosp, Coll Med, Seoul, South Korea Yonsei Univ, Songdang Inst Canc Res, Coll Med, Seoul, South Korea Yonsei Univ, Canc Prevent Ctr, Yonsei Canc Ctr, Coll Med, Seoul, South Korea
- [4] Discovery of dioxo-benzo[b]thiophene derivatives as potent YAP-TEAD interaction inhibitors for treating breast cancerBIOORGANIC CHEMISTRY, 2023, 131Son, Youngchai论文数: 0 引用数: 0 h-index: 0机构: Ewha Womans Univ, Coll Pharm, Seoul 03760, South Korea Ewha Womans Univ, Grad Sch Pharmaceut Sci, Seoul 03760, South Korea Korea Inst Sci & Technol KIST, Biomed Res Inst, Seoul 02792, South Korea Ewha Womans Univ, Coll Pharm, Seoul 03760, South KoreaKim, Jaeyeal论文数: 0 引用数: 0 h-index: 0机构: Korea Inst Sci & Technol KIST, Biomed Res Inst, Seoul 02792, South Korea Korea Univ, Dept Life Sci, Seoul 02841, South Korea Ewha Womans Univ, Coll Pharm, Seoul 03760, South KoreaKim, Yongchan论文数: 0 引用数: 0 h-index: 0机构: Korea Inst Sci & Technol KIST, Biomed Res Inst, Seoul 02792, South Korea Ewha Womans Univ, Coll Pharm, Seoul 03760, South KoreaChi, Sung -Gil论文数: 0 引用数: 0 h-index: 0机构: Korea Univ, Dept Life Sci, Seoul 02841, South Korea Ewha Womans Univ, Coll Pharm, Seoul 03760, South KoreaKim, Tackhoon论文数: 0 引用数: 0 h-index: 0机构: Korea Inst Sci & Technol KIST, Biomed Res Inst, Seoul 02792, South Korea Korea Univ, Dept Life Sci, Seoul 02841, South Korea Univ Sci & Technol, KIST Sch, Div Biomed Sci & Technol, Daejeon 34113, South Korea Ewha Womans Univ, Coll Pharm, Seoul 03760, South KoreaYu, Jinha论文数: 0 引用数: 0 h-index: 0机构: Ewha Womans Univ, Coll Pharm, Seoul 03760, South Korea Ewha Womans Univ, Grad Sch Pharmaceut Sci, Seoul 03760, South Korea Ewha Womans Univ, Coll Pharm, Seoul 03760, South Korea
- [5] Identification of small molecule Pan-TEAD inhibitors disrupting YAP-TEAD protein-protein interaction and targeting gastric cancer cellsCANCER RESEARCH, 2024, 84 (07)Kumar, Ramesh论文数: 0 引用数: 0 h-index: 0Toh, Joel论文数: 0 引用数: 0 h-index: 0Thian, Joanne论文数: 0 引用数: 0 h-index: 0Mohideen, Noorul Farzana论文数: 0 引用数: 0 h-index: 0Sun, Jialin论文数: 0 引用数: 0 h-index: 0Chakraborty, Sayan论文数: 0 引用数: 0 h-index: 0Gunaratne, Jayantha论文数: 0 引用数: 0 h-index: 0Hong, Wanjin论文数: 0 引用数: 0 h-index: 0
- [6] In vitro discovery of promising anti-cancer drug combinations using iterative maximisation of a therapeutic indexScientific Reports, 5M. Kashif论文数: 0 引用数: 0 h-index: 0机构: Uppsala University,C. Andersson论文数: 0 引用数: 0 h-index: 0机构: Uppsala University,S. Hassan论文数: 0 引用数: 0 h-index: 0机构: Uppsala University,H. Karlsson论文数: 0 引用数: 0 h-index: 0机构: Uppsala University,W. Senkowski论文数: 0 引用数: 0 h-index: 0机构: Uppsala University,M. Fryknäs论文数: 0 引用数: 0 h-index: 0机构: Uppsala University,P. Nygren论文数: 0 引用数: 0 h-index: 0机构: Uppsala University,R. Larsson论文数: 0 引用数: 0 h-index: 0机构: Uppsala University,M.G. Gustafsson论文数: 0 引用数: 0 h-index: 0机构: Uppsala University,
- [7] In vitro discovery of promising anti-cancer drug combinations using iterative maximisation of a therapeutic indexSCIENTIFIC REPORTS, 2015, 5Kashif, M.论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, Sweden Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, SwedenAndersson, C.论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, Sweden Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, SwedenHassan, S.论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, Sweden Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, SwedenKarlsson, H.论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, Sweden Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, SwedenSenkowski, W.论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, Sweden Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, SwedenFryknas, M.论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, Sweden Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, SwedenNygren, P.论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Immunol Genet & Pathol Expt & Clin Oncol, Akad Sjukhuset, SE-75185 Uppsala, Sweden Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, SwedenLarsson, R.论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, Sweden Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, SwedenGustafsson, M. G.论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, Sweden Uppsala Univ, Dept Med Sci Canc Pharmacol & Computat Med, Akad Sjukhuset, SE-75185 Uppsala, Sweden
- [8] Anti-cancer effects of glycogen synthase kinase 3 inhibitors discovered using structure-based drug discovery technologiesCANCER RESEARCH, 2009, 69Hyun, Young-Lan论文数: 0 引用数: 0 h-index: 0机构: CrystalGenomics Inc, Seoul, South Korea CrystalGenomics Inc, Seoul, South KoreaKim, Hyun Ji论文数: 0 引用数: 0 h-index: 0机构: CrystalGenomics Inc, Seoul, South Korea CrystalGenomics Inc, Seoul, South KoreaChoi, Eunha论文数: 0 引用数: 0 h-index: 0机构: CrystalGenomics Inc, Seoul, South Korea CrystalGenomics Inc, Seoul, South KoreaKim, Yong Eun论文数: 0 引用数: 0 h-index: 0机构: CrystalGenomics Inc, Seoul, South Korea CrystalGenomics Inc, Seoul, South KoreaLee, Dae Seung论文数: 0 引用数: 0 h-index: 0机构: CrystalGenomics Inc, Seoul, South Korea CrystalGenomics Inc, Seoul, South KoreaLee, Seung Chul论文数: 0 引用数: 0 h-index: 0机构: CrystalGenomics Inc, Seoul, South Korea CrystalGenomics Inc, Seoul, South KoreaPark, Myung Guan论文数: 0 引用数: 0 h-index: 0机构: CrystalGenomics Inc, Seoul, South Korea CrystalGenomics Inc, Seoul, South KoreaLee, Do Young论文数: 0 引用数: 0 h-index: 0机构: CrystalGenomics Inc, Seoul, South Korea CrystalGenomics Inc, Seoul, South KoreaChang, Ho-Jin论文数: 0 引用数: 0 h-index: 0机构: CrystalGenomics Inc, Seoul, South Korea CrystalGenomics Inc, Seoul, South KoreaChoi, Jong-Ryoo论文数: 0 引用数: 0 h-index: 0机构: CrystalGenomics Inc, Seoul, South Korea CrystalGenomics Inc, Seoul, South KoreaCho, Joong Myung论文数: 0 引用数: 0 h-index: 0机构: CrystalGenomics Inc, Seoul, South Korea CrystalGenomics Inc, Seoul, South KoreaRo, Seonggu论文数: 0 引用数: 0 h-index: 0机构: CrystalGenomics Inc, Seoul, South Korea CrystalGenomics Inc, Seoul, South Korea