2-Substituted Allyl Bromides as Electrophilic and Nucleophilic Building Blocks for 1,3-Dicarbonyl Compounds and Their Use in the Synthesis of Heterocycles

被引：0
作者：
Mineyeva, I., V [1 ]
机构：
[1] Belarusian State Univ, Minsk 220030, BELARUS
来源：
RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2022年 / 58卷 / 09期
关键词：
1; 3-dicarbonyl compounds; 2-substituted allyl bromides; methyl 3-(bromomethyl)but-3-enoate; 2-(bromomethyl)-4; 4-diethoxybut-1-ene; pyrazole; oxazole; benzo[f]coumarin; multicomponent reactions; COX-2; INHIBITORS; PART; DERIVATIVES; POTENT; ALDEHYDES; ETHYL;
D O I：
10.1134/S1070428022090032
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
An efficient procedure has been developed for the synthesis of new heterocyclic compounds from 2-substituted functionalized allyl bromides as precursors to electrophilic and nucleophilic building blocks for 1,3-dicarbonyl compounds.
引用
收藏
页码：1200 / 1212
页数：13
相关论文
共 40 条
  • [1] An Approach to the Synthesis of 2-Acylchromeno[3,4-c]pyrrol-4(2H)-one Derivatives via a Sequential Three-Component Reaction
    Alizadeh, Abdolali
    Ghanbaripour, Rashid
    Zhu, Long-Guan
    [J]. SYNLETT, 2013, 24 (16) : 2124 - 2126
  • [2] F(1H-Pyrazol-4-yl)methylene-Hydrazide derivatives: Synthesis and antimicrobial activity
    Bhavanarushi, Sangepu
    Luo, Zhi-Bin
    Bharath, Gandu
    Rani, JettiVatsala
    Khan, Imran
    Xu, Yin
    Liu, Bin
    Xie, Jimin
    [J]. JOURNAL OF HETEROCYCLIC CHEMISTRY, 2020, 57 (02) : 751 - 760
  • [3] The main directions and recent trends in the synthesis and use of isoxazoles
    Bondarenko, Oksana B.
    Zyk, Nikolai V.
    [J]. CHEMISTRY OF HETEROCYCLIC COMPOUNDS, 2020, 56 (06) : 694 - 707
  • [4] SYNTHESIS AND CHEMICAL-PROPERTIES OF PCA, AN UNUSUAL AMINO-ACID IN LUZOPEPTINS
    CIUFOLINI, MA
    XI, N
    [J]. JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1994, (16) : 1867 - 1868
  • [5] Cloricromene, a semi-synthetic coumarin derivative, inhibits tumor necrosis factor-α production at a pre-transcriptional level
    Corsini, E
    Lucchi, L
    Binaglia, M
    Viviani, B
    Bevilacqua, C
    Monastra, G
    Marinovich, M
    Galli, CL
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 2001, 418 (03) : 231 - 237
  • [6] Synthesis of a 2,3′;6′,3"-terpyridine scaffold as an α-helix mimetic
    Davis, JM
    Truong, A
    Hamilton, AD
    [J]. ORGANIC LETTERS, 2005, 7 (24) : 5405 - 5408
  • [7] Thermal, kinetic, spectroscopic studies and anti-microbial, anti-tuberculosis, anti-oxidant properties of clioquinol and benzo-coumarin derivatives mixed complexes with copper ion
    Dholariya, Hitesh R.
    Patel, Ketan S.
    Patel, Jiten C.
    Patel, Atul K.
    Patel, Kanuprasad D.
    [J]. MEDICINAL CHEMISTRY RESEARCH, 2013, 22 (12) : 5848 - 5860
  • [8] El-Ansary S. L., 1992, Egyptian Journal of Pharmaceutical Sciences, V33, P639
  • [9] Cannabinoid-1 receptor inverse agonists: current understanding of mechanism of action and unanswered questions
    Fong, T. M.
    Heymsfield, S. B.
    [J]. INTERNATIONAL JOURNAL OF OBESITY, 2009, 33 (09) : 947 - 955
  • [10] Design and synthesis of celecoxib and rofecoxib analogues as selective cyclooxygenase-2 (COX-2) inhibitors: Replacement of sulfonamide and methylsulfonyl pharmacophores by an azido bioisostere
    Habeeb, AG
    Rao, PNP
    Knaus, EE
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2001, 44 (18) : 3039 - 3042
1234