Synthesis of ML-3000, an inhibitor of cyclooxygenase and 5-lipoxygenase

被引：25

作者：

Cossy, J

Belotti, D

机构：

[1] Laboratoire de Chimie Organique, Associe au CNRS, ESPCI, 75231 Paris Cedex 05

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1997年 / 62卷 / 23期

关键词：

D O I：

10.1021/jo971480o

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：7900 / 7901

页数：2

共 11 条

[1] Reductive amination of aldehydes and ketones with sodium triacetoxyborohydride. Studies on direct and indirect reductive amination procedures [J].

AbdelMagid, AF ;

Carson, KG ;

Harris, BD ;

Maryanoff, CA ;

Shah, RD .

JOURNAL OF ORGANIC CHEMISTRY, 1996, 61 (11) :3849-3862

[2]

BELOTTI D, 1997, IN PRESS SYNLETT

[3] Cyclization of delta,epsilon-acetylenic amines and aminoacids into cyclic enamines. A very efficient and simple access to polysubstituted pyrrolidines. [J].

Cossy, J ;

Belotti, D ;

Bellosta, V ;

Boggio, C .

TETRAHEDRON LETTERS, 1997, 38 (15) :2677-2680

[4]

COSSY J, 1996, Patent No. 9612760

[5]

DIETL HK, 1973, TETRAHEDRON LETT, P1273

[6] SELECTIVE DEOXYGENATION OF KETONES AND ALDEHYDES INCLUDING HINDERED SYSTEMS WITH SODIUM CYANOBOROHYDRIDE [J].

HUTCHINS, RO ;

MILEWSKI, CA ;

MARYANOF.BE .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1973, 95 (11) :3662-3668

[7] (6,7-DIARYLDIHYDROPYRROLIZIN-5-YL)ACETIC ACIDS, A NOVEL CLASS OF POTENT DUAL INHIBITORS OF BOTH CYCLOOXYGENASE AND 5-LIPOXYGENASE [J].

LAUFER, SA ;

AUGUSTIN, J ;

DANNHARDT, G ;

KIEFER, W .

JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (12) :1894-1897

[8] PALLADIUM-CATALYZED CROSS-COUPLING REACTIONS OF ORGANOBORON COMPOUNDS [J].

MIYAURA, N ;

SUZUKI, A .

CHEMICAL REVIEWS, 1995, 95 (07) :2457-2483

[9]

Rabasseda X., 1995, Drugs of the Future, V20, P1007

[10]

RITTER K, 1993, SYNTHESIS-STUTTGART, P735

← 1 2 →