Alanine scanning of VIP -: Structure-function relationship for binding to human recombinant VPAC1 receptor

被引：0
|
作者：
Nicole, P
Rouyer-Fessard, C
Couvineau, A
Drouot, C
Fulcrand, P
Martinez, J
Laburthe, M [1 ]
机构：
[1] Fac Med Bichat, INSERM, U410, F-75018 Paris, France
[2] CNRS, URM5810, F-34094 Montpellier, France
来源：
VIP, PACAP, GLUCAGON, AND RELATED PEPTIDES | 2000年 / 921卷
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：352 / 356
页数：5
相关论文
共 50 条
  • [1] Tryptophan 67 in the human VPAC1 receptor:: Crucial role for VIP binding
    Nicole, P
    Maoret, JJ
    Couvineau, A
    Momany, FA
    Laburthe, M
    BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2000, 276 (02) : 654 - 659
  • [2] Alanine-scanning of VIP and molecular modeling of VIP analogs: Determination of important residues for interaction with human VPAC1 and VPAC2 receptors
    Laburthe, M
    Nicole, P
    Rouyer-Fessard, C
    Couvineau, A
    Maoret, JJ
    Drouot, C
    Fulcrand, P
    Martinez, J
    Lins, L
    Thomas, A
    Brasseur, R
    GASTROENTEROLOGY, 1999, 116 (04) : A621 - A621
  • [3] VPAC1 receptor: identification of different binding sites of VIP and an antagonist by photolabeling and modeling
    Ceraudo, Emilie
    Tan, Yossan-Var
    Nicole, Pascal
    Couvineau, Alain
    Laburthe, Marc
    JOURNAL OF MOLECULAR NEUROSCIENCE, 2010, 42 (03) : 313 - 313
  • [4] Elucidation of the VIP pharmacophore for human VPAC1 and VPAC2 and development of simplified VIP analogs with receptor selectivity and stability
    Igarashi, Hisato
    Ito, Tetsuhide
    Yoshinaga, Masahiro
    Sakai, Hironori
    Muto, Yoichi
    Takayanagi, Ryoichi
    Coy, David H.
    Jensen, Robert T.
    REGULATORY PEPTIDES, 2006, 135 (03) : 131 - 131
  • [5] Demonstration of physical interactions between VIP and the N-terminal ectodomain of human VPAC1 receptor by photoaffinity scanning
    Tan, YV
    Couvineau, A
    Laburthe, M
    REGULATORY PEPTIDES, 2004, 122 (01) : 42 - 42
  • [6] Identification of key residues for interaction of vasoactive intestinal peptide with human VPAC1 and VPAC2 receptors and development of a highly selective VPAC1 receptor agonist -: Alanine scanning and molecular modeling of the peptide
    Nicole, P
    Lins, L
    Rouyer-Fessard, C
    Drouot, C
    Fulcrand, P
    Thomas, A
    Couvineau, A
    Martinez, J
    Brasseur, R
    Laburthe, M
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2000, 275 (31) : 24003 - 24012
  • [7] In Silico Classification and Prediction of VIP Derivatives as VPAC1/VPAC2 Receptor Agonists/Antagonists
    Li, Jiazhong
    Wang, Xin
    Liu, Huanxiang
    Li, Hongyu
    COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING, 2015, 18 (01) : 33 - 41
  • [8] Internalization and trafficking of the VIP receptors:: A comparison between the recombinant VPAC1 and VPAC2 human receptors expressed in cho cells
    Langlet, C
    Gaspard, N
    Vertongen, P
    Robberecht, P
    Langer, I
    REGULATORY PEPTIDES, 2004, 122 (01) : 26 - 26
  • [9] STRUCTURE-FUNCTION RELATIONSHIP OF A RECOMBINANT HUMAN GALACTOSIDE-BINDING PROTEIN
    OCHIENG, J
    PLATT, D
    TAIT, L
    HOGAN, V
    RAZ, T
    CARMI, P
    RAZ, A
    BIOCHEMISTRY, 1993, 32 (16) : 4455 - 4460
  • [10] Vasoactive intestinal polypeptide (VIP) and VPAC1 receptor in adult human dental pulp in relation to caries
    El Karim, Ikhlas A.
    Lamey, Philip-John
    Ardill, Joy
    Linden, Gerard J.
    Lundy, Fionnuala T.
    ARCHIVES OF ORAL BIOLOGY, 2006, 51 (10) : 849 - 855
12345