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- [23] Synthesis and Pharmacological Characterization of C4β-Amide-Substituted 2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylates. Identification of (1S,2S,4S,5R,6S)-2-Amino-4-[(3-methoxybenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic Acid (LY2794193), a Highly Potent and Selective mGlu3 Receptor Agonist JOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (06) : 2303 - 2328
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- [29] Use of silyl ester and enamine protection for an efficient alternate synthesis of (1S,2S,5R,6S)-2-[(2′S)-(2′-amino)propionyl]aminobicyclo[3.1.0] hexane-2,6-dicarboxylic acid hydrochloride (LY544344•HCl) SYNTHESIS-STUTTGART, 2006, (16): : 2659 - 2664