Synthesis and insecticidal activity of fluorinated 2-(2,6-dichloro-4-trifluoromethylphenyl)-2,4,5,6-tetrahydrocyclopentapyrazoles

被引:13
作者
Meegalla, SK
Doller, D
Liu, RP
Sha, DY
Lee, Y
Soll, RM
Wisnewski, N
Silver, GM
Dhanoa, D
机构
[1] Johnson & Johnson Pharmaceut Res & Dev, Exton, PA 19341 USA
[2] Heska Corp, Ft Collins, CO 80525 USA
关键词
phenylpyrazole; GABA; fipronil; anti-flea; anti-tick;
D O I
10.1016/j.bmcl.2005.12.012
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
A number of fluorinated 1-aryl-tetrahydrocyclopentapyrazoles were synthesized and their insecticidal activity was evaluated. Some of the fluorinated compounds had significant insecticidal properties. (C) 2005 Elsevier Ltd. All rights reserved.
引用
收藏
页码:1702 / 1706
页数:5
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Meegalla, SK ;
Doller, D ;
Liu, RP ;
Sha, DY ;
Soll, RM ;
Dhanoa, DS .
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[3]  
Olah G. A., 1992, SYNTHETIC FLUORINE C