共 15 条
Advances at the intersection of chemical biology and medicinal chemistry
被引:2
作者:

论文数: 引用数:
h-index:
机构:
机构:
[1] Univ Southampton, Southampton SO17 1RE, Hants, England
关键词:
chemical biology;
drug design;
drug discovery;
medicinal chemistry;
D O I:
10.4155/fmc.15.151
中图分类号:
R914 [药物化学];
学科分类号:
100701 ;
摘要:
引用
收藏
页码:2089 / 2090
页数:2
相关论文
共 15 条
[1]
Beyond cyclosporine A: conformation-dependent passive membrane permeabilities of cyclic peptide natural products
[J].
Ahlbach, Christopher L.
;
Lexa, Katrina W.
;
Bockus, Andrew T.
;
Chen, Valerie
;
Crews, Phillip
;
Jacobson, Matthew P.
;
Lokey, R. Scott
.
FUTURE MEDICINAL CHEMISTRY,
2015, 7 (16)
:2121-2130

Ahlbach, Christopher L.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif Santa Cruz, Dept Chem & Biochem, Santa Cruz, CA 95064 USA Univ Calif Santa Cruz, Dept Chem & Biochem, Santa Cruz, CA 95064 USA

Lexa, Katrina W.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Dept Pharmaceut Chem, San Francisco, CA 94158 USA Univ Calif Santa Cruz, Dept Chem & Biochem, Santa Cruz, CA 95064 USA

Bockus, Andrew T.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif Santa Cruz, Dept Chem & Biochem, Santa Cruz, CA 95064 USA Univ Calif Santa Cruz, Dept Chem & Biochem, Santa Cruz, CA 95064 USA

Chen, Valerie
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif Santa Cruz, Dept Chem & Biochem, Santa Cruz, CA 95064 USA Univ Calif Santa Cruz, Dept Chem & Biochem, Santa Cruz, CA 95064 USA

Crews, Phillip
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif Santa Cruz, Dept Chem & Biochem, Santa Cruz, CA 95064 USA Univ Calif Santa Cruz, Dept Chem & Biochem, Santa Cruz, CA 95064 USA

Jacobson, Matthew P.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Dept Pharmaceut Chem, San Francisco, CA 94158 USA Univ Calif Santa Cruz, Dept Chem & Biochem, Santa Cruz, CA 95064 USA

Lokey, R. Scott
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif Santa Cruz, Dept Chem & Biochem, Santa Cruz, CA 95064 USA Univ Calif Santa Cruz, Dept Chem & Biochem, Santa Cruz, CA 95064 USA
[2]
Sialic acids in biological and therapeutic processes: opportunities and challenges
[J].
Bauer, Julia
;
Osborn, Helen M. I.
.
FUTURE MEDICINAL CHEMISTRY,
2015, 7 (16)
:2285-2299

Bauer, Julia
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Reading, Reading Sch Pharm, Reading RG6 6AD, Berks, England Univ Reading, Reading Sch Pharm, Reading RG6 6AD, Berks, England

Osborn, Helen M. I.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Reading, Reading Sch Pharm, Reading RG6 6AD, Berks, England Univ Reading, Reading Sch Pharm, Reading RG6 6AD, Berks, England
[3]
Rational approach to an antiprion compound with a multiple mechanism of action
[J].
Bolognesi, Maria Laura
;
Bongarzone, Salvatore
;
Aulic, Suzana
;
Hoang Ngoc Ai Tran
;
Prati, Federica
;
Carloni, Paolo
;
Legname, Giuseppe
.
FUTURE MEDICINAL CHEMISTRY,
2015, 7 (16)
:2113-2120

Bolognesi, Maria Laura
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Bologna, Dept Pharm & Biotechnol, Alma Mater Studiorum, I-40126 Bologna, Italy Univ Bologna, Dept Pharm & Biotechnol, Alma Mater Studiorum, I-40126 Bologna, Italy

Bongarzone, Salvatore
论文数: 0 引用数: 0
h-index: 0
机构:
St Thomas Hosp, Kings Coll London, Div Imaging Sci & Biomed Engn, Kings Hlth Partners, London SE1 7EH, England Univ Bologna, Dept Pharm & Biotechnol, Alma Mater Studiorum, I-40126 Bologna, Italy

Aulic, Suzana
论文数: 0 引用数: 0
h-index: 0
机构:
SISSA, Dept Neurosci, I-34136 Trieste, Italy Univ Bologna, Dept Pharm & Biotechnol, Alma Mater Studiorum, I-40126 Bologna, Italy

Hoang Ngoc Ai Tran
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calgary, Dept Comparat & Biol Expt Med, Calgary, AB, Canada Univ Bologna, Dept Pharm & Biotechnol, Alma Mater Studiorum, I-40126 Bologna, Italy

Prati, Federica
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Bologna, Dept Pharm & Biotechnol, Alma Mater Studiorum, I-40126 Bologna, Italy Univ Bologna, Dept Pharm & Biotechnol, Alma Mater Studiorum, I-40126 Bologna, Italy

Carloni, Paolo
论文数: 0 引用数: 0
h-index: 0
机构:
Inst Adv Simulat, Computat Biomed Sect IAS 5, D-52425 Julich, Germany
Julich RWTH Aachen, Lab Computat Biophys, German Res Sch Simulat Sci GRS, Julich, Germany Univ Bologna, Dept Pharm & Biotechnol, Alma Mater Studiorum, I-40126 Bologna, Italy

Legname, Giuseppe
论文数: 0 引用数: 0
h-index: 0
机构:
SISSA, Dept Neurosci, I-34136 Trieste, Italy Univ Bologna, Dept Pharm & Biotechnol, Alma Mater Studiorum, I-40126 Bologna, Italy
[4]
Rational, computer-enabled peptide drug design: principles, methods, applications and future directions
[J].
Diller, David J.
;
Swanson, Jon
;
Bayden, Alexander S.
;
Jarosinski, Mark
;
Audie, Joseph
.
FUTURE MEDICINAL CHEMISTRY,
2015, 7 (16)
:2173-2193

Diller, David J.
论文数: 0 引用数: 0
h-index: 0
机构:
CMD Biosci, New Haven, CT 06511 USA CMD Biosci, New Haven, CT 06511 USA

Swanson, Jon
论文数: 0 引用数: 0
h-index: 0
机构:
ChemModeling LLC, Weldon Spring, MO 63304 USA CMD Biosci, New Haven, CT 06511 USA

Bayden, Alexander S.
论文数: 0 引用数: 0
h-index: 0
机构:
CMD Biosci, New Haven, CT 06511 USA CMD Biosci, New Haven, CT 06511 USA

Jarosinski, Mark
论文数: 0 引用数: 0
h-index: 0
机构:
CMD Biosci, New Haven, CT 06511 USA CMD Biosci, New Haven, CT 06511 USA

Audie, Joseph
论文数: 0 引用数: 0
h-index: 0
机构:
CMD Biosci, New Haven, CT 06511 USA
Sacred Heart Univ, Dept Chem, Fairfield, CT 06825 USA CMD Biosci, New Haven, CT 06511 USA
[5]
Cell permeable affinity- and activity-based probes
[J].
Jones, Lyn H.
.
FUTURE MEDICINAL CHEMISTRY,
2015, 7 (16)
:2131-2141

Jones, Lyn H.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer, WorldWide Med Chem, Cambridge, MA 02139 USA Pfizer, WorldWide Med Chem, Cambridge, MA 02139 USA
[6]
Successful strategies in the discovery of small-molecule epigenetic modulators with anticancer potential
[J].
Juan Bayo
;
Dalvi, Maithili P.
;
Martinez, Elisabeth D.
.
FUTURE MEDICINAL CHEMISTRY,
2015, 7 (16)
:2243-2261

Juan Bayo
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Texas SW Med Ctr Dallas, Dept Pharmacol, Dallas, TX 75390 USA Univ Texas SW Med Ctr Dallas, Dept Pharmacol, Dallas, TX 75390 USA

Dalvi, Maithili P.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Texas SW Med Ctr Dallas, Hamon Ctr Therapeut Oncol Res, Dallas, TX 75390 USA Univ Texas SW Med Ctr Dallas, Dept Pharmacol, Dallas, TX 75390 USA

Martinez, Elisabeth D.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Texas SW Med Ctr Dallas, Dept Pharmacol, Dallas, TX 75390 USA
Univ Texas SW Med Ctr Dallas, Hamon Ctr Therapeut Oncol Res, Dallas, TX 75390 USA Univ Texas SW Med Ctr Dallas, Dept Pharmacol, Dallas, TX 75390 USA
[7]
Recent developments and applications of clickable photoprobes in medicinal chemistry and chemical biology
[J].
Lapinsky, David J.
;
Johnson, Douglas S.
.
FUTURE MEDICINAL CHEMISTRY,
2015, 7 (16)
:2143-2171

Lapinsky, David J.
论文数: 0 引用数: 0
h-index: 0
机构:
Duquesne Univ, Div Pharmaceut Sci, Pittsburgh, PA 15282 USA Duquesne Univ, Div Pharmaceut Sci, Pittsburgh, PA 15282 USA

Johnson, Douglas S.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Neurosci Med Chem & Chem Biol, Cambridge, MA 02139 USA Duquesne Univ, Div Pharmaceut Sci, Pittsburgh, PA 15282 USA
[8]
Targeting cell death pathways with small molecules: playing with life and death at the cellular level to treat diseases
[J].
Lessene, Guillaume
.
FUTURE MEDICINAL CHEMISTRY,
2015, 7 (16)
:2099-2102

Lessene, Guillaume
论文数: 0 引用数: 0
h-index: 0
机构:
Walter & Eliza Hall Inst Med Res, ACRF Chem Biol Div, Parkville, Vic 3052, Australia
Univ Melbourne, Dept Med Biol, Melbourne, Vic 3050, Australia
Univ Melbourne, Dept Pharmacol & Therapeut, Melbourne, Vic 3050, Australia Walter & Eliza Hall Inst Med Res, ACRF Chem Biol Div, Parkville, Vic 3052, Australia
[9]
Toward peptide-based inhibitors as therapies for Parkinson's disease
[J].
Mason, Jody M.
;
Fairlie, David P.
.
FUTURE MEDICINAL CHEMISTRY,
2015, 7 (16)
:2103-2105

Mason, Jody M.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Bath, Dept Biol & Biochem, Bath BA2 7AY, Avon, England Univ Bath, Dept Biol & Biochem, Bath BA2 7AY, Avon, England

Fairlie, David P.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Queensland, Inst Mol Biosci, Div Chem & Struct Biol, Brisbane, Qld, Australia Univ Bath, Dept Biol & Biochem, Bath BA2 7AY, Avon, England
[10]
Harnessing dynamic combinatorial chemistry in the search for new ligands for protein targets
[J].
Monjas, Leticia
;
Hirsch, Anna K. H.
.
FUTURE MEDICINAL CHEMISTRY,
2015, 7 (16)
:2095-2098

论文数: 引用数:
h-index:
机构:

Hirsch, Anna K. H.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Groningen, Stratingh Inst Chem, NL-9747 AG Groningen, Netherlands Univ Groningen, Stratingh Inst Chem, NL-9747 AG Groningen, Netherlands