Inhibition of imatinib transport by uremic toxins during renal failure

被引:15
作者
Franke, Ryan M. [1 ]
Sparreboom, Alex [1 ]
机构
[1] St Jude Childrens Hosp, Dept Pharmaceut Sci, Memphis, TN 38105 USA
关键词
D O I
10.1200/JCO.2008.18.4390
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:4226 / 4227
页数:3
相关论文
共 16 条
[1]  
Gelderblom H, 1999, DRUG METAB DISPOS, V27, P1300
[2]   Phase I and pharmacokinetic study of imatinib mesylate in patients with advanced malignancies and varying degrees of renal dysfunction: A study by the National Cancer Institute Organ Dysfunction Working Group [J].
Gibbons, Joseph ;
Egorin, Merrill J. ;
Ramanathan, Ramesh K. ;
Fu, Pingfu ;
Mulkerin, Daniel L. ;
Shibata, Stephen ;
Takimoto, Chris H. M. ;
Mani, Sridhar ;
LoRusso, Patricia A. ;
Grem, Jean L. ;
Pavlick, Anna ;
Lenz, Heinz-Josef ;
Flick, Susan M. ;
Reynolds, Sherrie ;
Lagattuta, Theodore F. ;
Parise, Robert A. ;
Wang, Yanfeng ;
Murgo, Anthony J. ;
Ivy, S. Percy ;
Remick, Scot C. .
JOURNAL OF CLINICAL ONCOLOGY, 2008, 26 (04) :570-576
[3]  
HENDERSON SJ, 1992, J PHARMACOL EXP THER, V263, P54
[4]   Interaction of imatinib with human organic ion carriers [J].
Hu, Shuiying ;
Franke, Ryan M. ;
Filipski, Kelly K. ;
Hu, Chaoxin ;
Orwick, Shelley J. ;
de Bruijn, Ernst A. ;
Burger, Herman ;
Baker, Sharyn D. ;
Sparreboom, Alex .
CLINICAL CANCER RESEARCH, 2008, 14 (10) :3141-3148
[5]   Imatinib for patients with liver or kidney dysfunction: No need to modify the dose [J].
Judson, Ian R. .
JOURNAL OF CLINICAL ONCOLOGY, 2008, 26 (04) :521-522
[6]  
Leblond F, 2001, J AM SOC NEPHROL, V12, P326, DOI 10.1681/ASN.V122326
[7]   Downregulation of intestinal cytochrome P450 in chronic renal failure [J].
Leblond, FA ;
Petrucci, M ;
Dubé, P ;
Bernier, G ;
Bonnardeaux, A ;
Pichette, V .
JOURNAL OF THE AMERICAN SOCIETY OF NEPHROLOGY, 2002, 13 (06) :1579-1585
[8]   A FURAN FATTY-ACID AND INDOXYL SULFATE ARE THE PUTATIVE INHIBITORS OF THYROXINE HEPATOCYTE TRANSPORT IN UREMIA [J].
LIM, CF ;
BERNARD, BF ;
DEJONG, M ;
DOCTER, R ;
KRENNING, EP ;
HENNEMANN, G .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1993, 76 (02) :318-324
[9]  
NIWA T, 1994, J LAB CLIN MED, V124, P96
[10]  
NIWA T, 1993, CLIN NEPHROL, V39, P92