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- [29] The Discovery of (S)-1-(6-(34(4-(1-(Cyclopropanecarbonyl)piperidin-4-y1)-2-methylphenypamino)-2,3-dihydro-1H-inden-4-yl)pyridin-2-yl)-5-methyl-1H-pyrazole-4-carboxylic Acid, a Soluble Guanylate Cyclase Activator Specifically Designed for Topical Ocular Delivery as a Therapy for Glaucoma JOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (06) : 2552 - 2570