Thromboxane (A2) receptor antagonists as potential candidates for Alzheimer's disease

被引:0
作者
Ballatore, Carlo [1 ]
Herbst-Robinson, Katie [2 ]
Wang, Xiaozhao [1 ]
Soper, James H. [2 ]
Sugiyama, Shimpei [1 ]
James, Michael J. [2 ]
Huang, Longchuan [1 ]
Yao, Mandy [2 ]
Lee, Virginia M. -Y. [2 ]
Trojanowski, John Q. [2 ]
Brunden, Kurt R. [2 ]
Smith, Amos B., III [1 ]
机构
[1] Univ Penn, Dept Chem, Philadelphia, PA 19104 USA
[2] Univ Penn, Dept Pathol & Lab Med, Philadelphia, PA 19104 USA
来源
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2013年 / 245卷
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
267-MEDI
引用
收藏
页数:1
相关论文
共 50 条
[41]   SYNTHETIC THROMBOXANE-A2 AND CHARACTERIZATION OF THE THROMBOXANE RECEPTOR USING A NOVEL CLASS OF RECEPTOR ANTAGONISTS [J].
MORTON, HE ;
EVANS, J ;
LEVEILLE, C ;
LORD, A ;
GILLARD, JW .
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1988, 195 :122-MEDI
[42]   Pathophysiological Role and Medicinal Chemistry of A2A Adenosine Receptor Antagonists in Alzheimer's Disease [J].
Merighi, Stefania ;
Borea, Pier Andrea ;
Varani, Katia ;
Vincenzi, Fabrizio ;
Travagli, Alessia ;
Nigro, Manuela ;
Pasquini, Silvia ;
Suresh, R. Rama ;
Kim, Sung Won ;
Volkow, Nora D. ;
Jacobson, Kenneth A. ;
Gessi, Stefania .
MOLECULES, 2022, 27 (09)
[43]   Angiotensin II Type 1 (AT1) receptor antagonists as potential candidates for anxiety treatment in Parkinson's Disease [J].
Bordet, S. ;
Grasso, L. ;
Udovin, L. ;
Chevalier, G. ;
Otero-Losada, M. ;
Capani, F. ;
Perez-Lloret, S. .
MOVEMENT DISORDERS, 2023, 38 :S599-S602
[44]   Phospholipase A2 and arachidonic acid in Alzheimer's disease [J].
Sanchez-Mejia, Rene O. ;
Mucke, Lennart .
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR AND CELL BIOLOGY OF LIPIDS, 2010, 1801 (08) :784-790
[45]   The β1-Subunit of the MaxiK Channel Associates with the Thromboxane A2 Receptor and Reduces Thromboxane A2 Functional Effects [J].
Li, Min ;
Zhang, Zhu ;
Koh, Huilin ;
Lu, Rong ;
Jiang, Zhaorong ;
Alioua, Abderrahmane ;
Garcia-Valdes, Jesus ;
Stefani, Enrico ;
Toro, Ligia .
JOURNAL OF BIOLOGICAL CHEMISTRY, 2013, 288 (05) :3668-3677
[46]   Transient receptor potential channels in Alzheimer's disease [J].
Yamamoto, Shinichiro ;
Wajima, Teruaki ;
Hara, Yuji ;
Nishida, Motohiro ;
Mori, Yasuo .
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR BASIS OF DISEASE, 2007, 1772 (08) :958-967
[47]   Protection of atherogenesis in thromboxane A2 receptor-deficient mice is not associated with thromboxane A2 receptor in bone marrow-derived cells [J].
Zhuge, Xin ;
Arai, Hidenori ;
Xu, Yang ;
Murayama, Toshinorl ;
Kobayashi, Takuya ;
Narumiya, Shuh ;
Kita, Toru ;
Yokode, Masayuki .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2006, 351 (04) :865-871
[48]   Synthesis and pharmacological evaluation of 2-aryloxy/arylamino-5-cyanobenzenesulfonylureas as novel thromboxane A2 receptor antagonists [J].
Bambi-Nyanguile, Sylvie-Mireille ;
Hanson, Julien ;
Ooms, Annie ;
Alpan, Lutfiye ;
Kolh, Philippe ;
Dogne, Jean-Michel ;
Pirotte, Bernard .
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 65 :32-40
[49]   MEDI 267-Development of dual-acting benzofurans and benzomorpholines as thromboxane A2 receptor antagonists and prostacyclin receptor agonists [J].
Ohno, Michihiro ;
Miyamoto, Mitsuko ;
Takeda, Takahiro ;
Tanaka, Yoichiro ;
Makita, Kei ;
Hoshi, Kazuhiro ;
Yamada, Naohiro ;
Ohtake, Atsushi .
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2006, 232
[50]   SYNTHESIS OF THROMBOXANE RECEPTOR ANTAGONISTS WITH THE POTENTIAL TO RADIOLABEL WITH I-125 [J].
MAIS, D ;
KNAPP, D ;
HALUSHKA, P ;
BALLARD, K ;
HAMANAKA, N .
TETRAHEDRON LETTERS, 1984, 25 (38) :4207-4210