Brine-Mediated Efficient Benzoylation of Primary Amines and Amino Acids

被引：15

作者：

Chattopadhyay, Gautam ^{[1
]}

Chakraborty, Suchandra ^{[2
]}

Saha, Chandan ^{[2
]}

机构：

[1] Presidency Coll, Postgrad Dept Chem, Kolkata 700073, W Bengal, India

[2] Sch Trop Med, Dept Clin & Expt Pharmacol, Kolkata, India

来源：

SYNTHETIC COMMUNICATIONS | 2008年 / 38卷 / 23期

关键词：

Amines; amino acids; benzoylation; brine;

D O I：

10.1080/00397910802250929

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Benzoylation of primary amines and amino acids is efficiently carried out in a brine solution using a stoichiometric amount of benzoyl chloride followed by trituration with aqueous saturated bicarbonate solution.

引用

页码：4068 / 4075

页数：8

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