Synthetic study on hapalosin, a cyclic depsipeptide possessing multidrug resistance reversing activities

被引：25

作者：

Ohmori, K ^{[1
]}

Okuno, T ^{[1
]}

Nishiyama, S ^{[1
]}

Yamamura, S ^{[1
]}

机构：

[1] KEIO UNIV,FAC SCI & TECHNOL,DEPT CHEM,YOKOHAMA 223,JAPAN

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 20期

关键词：

D O I：

10.1016/0040-4039(96)00592-8

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Hapalosin possessing a multidrug resistance reversing activity, has been synthesized from the corresponding hydroxy acids and gamma-amino acids. The stereochemistry of the natural product and related derivatives is discussed. Copyright (C) 1996 Elsevier Science Ltd

引用

页码：3467 / 3470

页数：4

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