首页
学术期刊
论文检测
AIGC检测
热点
更多
数据
Practical synthesis and SAR study of aliskiren: An orally active human renin inhibitor
被引:0
|
作者
:
Dong, Hua
论文数:
0
引用数:
0
h-index:
0
机构:
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
Dong, Hua
[
1
]
Zhang, Zhi-Liu
论文数:
0
引用数:
0
h-index:
0
机构:
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
Zhang, Zhi-Liu
[
1
]
Huang, Lia-Hui
论文数:
0
引用数:
0
h-index:
0
机构:
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
Huang, Lia-Hui
[
1
]
Ma, Rujian
论文数:
0
引用数:
0
h-index:
0
机构:
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
Ma, Rujian
[
1
]
Chen, Shu-Hui
论文数:
0
引用数:
0
h-index:
0
机构:
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
Chen, Shu-Hui
[
1
]
Li, Ge
论文数:
0
引用数:
0
h-index:
0
机构:
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
Li, Ge
[
1
]
机构
:
[1]
WuXi PharmaTech Co Ltd, Shanghai 200131, Peoples R China
来源
:
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY
|
2005年
/ 230卷
关键词
:
D O I
:
暂无
中图分类号
:
O6 [化学];
学科分类号
:
0703 ;
摘要
:
341-MEDI
引用
收藏
页码:U2696 / U2696
页数:1
相关论文
共 50 条
[21]
Pharmacokinetics of remikiren, a potent orally active inhibitor of human renin, in rat, dog and primates
Coassolo, P
论文数:
0
引用数:
0
h-index:
0
机构:
Pharma Division Preclinical Research, F. Hoffmann-La Roche AG
Coassolo, P
Fischli, W
论文数:
0
引用数:
0
h-index:
0
机构:
Pharma Division Preclinical Research, F. Hoffmann-La Roche AG
Fischli, W
Clozel, JP
论文数:
0
引用数:
0
h-index:
0
机构:
Pharma Division Preclinical Research, F. Hoffmann-La Roche AG
Clozel, JP
Chou, RC
论文数:
0
引用数:
0
h-index:
0
机构:
Pharma Division Preclinical Research, F. Hoffmann-La Roche AG
Chou, RC
XENOBIOTICA,
1996,
26
(03)
: 333
-
345
[22]
Aliskiren, an orally effective renin inhibitor, shows dose linear pharmacokinetics in healthy volunteers.
Vaidyanathan, S
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Pharmaceut, E Hanover, NJ USA
Vaidyanathan, S
Limoges, D
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Pharmaceut, E Hanover, NJ USA
Limoges, D
Yeh, C
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Pharmaceut, E Hanover, NJ USA
Yeh, C
Dieterich, H
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Pharmaceut, E Hanover, NJ USA
Dieterich, H
CLINICAL PHARMACOLOGY & THERAPEUTICS,
2006,
79
(02)
: P64
-
P64
[23]
Suppression of the renin system by the novel orally effective direct renin inhibitor aliskiren: A pooled analysis of 1612 patients with hypertension
Gradman, Alan H.
论文数:
0
引用数:
0
h-index:
0
机构:
Western Penn Hosp, Pittsburgh, PA 15224 USA
Gradman, Alan H.
Flack, John M.
论文数:
0
引用数:
0
h-index:
0
机构:
Western Penn Hosp, Pittsburgh, PA 15224 USA
Flack, John M.
Arora, Vipin
论文数:
0
引用数:
0
h-index:
0
机构:
Western Penn Hosp, Pittsburgh, PA 15224 USA
Arora, Vipin
Zhang, Jack
论文数:
0
引用数:
0
h-index:
0
机构:
Western Penn Hosp, Pittsburgh, PA 15224 USA
Zhang, Jack
Anderson, David R.
论文数:
0
引用数:
0
h-index:
0
机构:
Western Penn Hosp, Pittsburgh, PA 15224 USA
Anderson, David R.
Keefe, Deborah L.
论文数:
0
引用数:
0
h-index:
0
机构:
Western Penn Hosp, Pittsburgh, PA 15224 USA
Keefe, Deborah L.
Satlin, Andrew
论文数:
0
引用数:
0
h-index:
0
机构:
Western Penn Hosp, Pittsburgh, PA 15224 USA
Satlin, Andrew
Prescott, Margaret F.
论文数:
0
引用数:
0
h-index:
0
机构:
Western Penn Hosp, Pittsburgh, PA 15224 USA
Prescott, Margaret F.
CIRCULATION,
2006,
114
(18)
: 773
-
773
[24]
Total Synthesis of "Aliskiren": The First Renin Inhibitor in Clinical Practice for Hypertension
Hanessian, Stephen
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Montreal, Dept Chem, Montreal, PQ H3C 3J7, Canada
Univ Montreal, Dept Chem, Montreal, PQ H3C 3J7, Canada
Hanessian, Stephen
Guesne, Sebastien
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Montreal, Dept Chem, Montreal, PQ H3C 3J7, Canada
Univ Montreal, Dept Chem, Montreal, PQ H3C 3J7, Canada
Guesne, Sebastien
Chenard, Etienne
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Montreal, Dept Chem, Montreal, PQ H3C 3J7, Canada
Univ Montreal, Dept Chem, Montreal, PQ H3C 3J7, Canada
Chenard, Etienne
ORGANIC LETTERS,
2010,
12
(08)
: 1816
-
1819
[25]
Aliskiren, a novel orally effective renin inhibitor, exhibits similar pharmacokinetics and pharmacodynamics in Japanese and Caucasian subjects
Vaidyanathan, S
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis, Exploratory Clin Dev, E Hanover, NJ USA
Novartis, Exploratory Clin Dev, E Hanover, NJ USA
Vaidyanathan, S
Jermany, J
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis, Exploratory Clin Dev, E Hanover, NJ USA
Novartis, Exploratory Clin Dev, E Hanover, NJ USA
Jermany, J
Yeh, CM
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis, Exploratory Clin Dev, E Hanover, NJ USA
Novartis, Exploratory Clin Dev, E Hanover, NJ USA
Yeh, CM
Bizot, MN
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis, Exploratory Clin Dev, E Hanover, NJ USA
Novartis, Exploratory Clin Dev, E Hanover, NJ USA
Bizot, MN
Camisasca, RP
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis, Exploratory Clin Dev, E Hanover, NJ USA
Novartis, Exploratory Clin Dev, E Hanover, NJ USA
Camisasca, RP
AMERICAN JOURNAL OF HYPERTENSION,
2005,
18
(05)
: 75A
-
76A
[26]
Aliskiren, a novel, orally effective renin inhibitor, lowers blood pressure in marmosets and spontaneously hypertensive rats
Wood, JM
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Inst BioMed Res, E Hanover, NJ 07936 USA
Wood, JM
Schnell, CR
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Inst BioMed Res, E Hanover, NJ 07936 USA
Schnell, CR
Cumin, F
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Inst BioMed Res, E Hanover, NJ 07936 USA
Cumin, F
Menard, J
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Inst BioMed Res, E Hanover, NJ 07936 USA
Menard, J
Webb, RL
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Inst BioMed Res, E Hanover, NJ 07936 USA
Webb, RL
JOURNAL OF HYPERTENSION,
2005,
23
(02)
: 417
-
426
[27]
Aliskiren, a novel orally effective renin inhibitor, exhibits similar pharmacokinetics and pharmacodynamics in Japanese and Caucasian subjects
Vaidyanathan, Sujata
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Pharmaceut, E Hanover, NJ 07936 USA
Novartis Pharmaceut, E Hanover, NJ 07936 USA
Vaidyanathan, Sujata
Jermany, Joanne
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Pharmaceut, E Hanover, NJ 07936 USA
Jermany, Joanne
Yeh, ChingMing
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Pharmaceut, E Hanover, NJ 07936 USA
Yeh, ChingMing
Bizot, Marie-Noelle
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Pharmaceut, E Hanover, NJ 07936 USA
Bizot, Marie-Noelle
Camisasca, Riccardo
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Pharmaceut, E Hanover, NJ 07936 USA
Camisasca, Riccardo
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY,
2006,
62
(06)
: 690
-
698
[28]
First experience with an orally active benin inhibitor (aliskiren) in patients with chronic heart failure
Seed, A
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Glasgow, Glasgow G12 8QQ, Lanark, Scotland
Seed, A
Gardner, R
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Glasgow, Glasgow G12 8QQ, Lanark, Scotland
Gardner, R
McMurray, J
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Glasgow, Glasgow G12 8QQ, Lanark, Scotland
McMurray, J
Hillier, C
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Glasgow, Glasgow G12 8QQ, Lanark, Scotland
Hillier, C
Murdoch, D
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Glasgow, Glasgow G12 8QQ, Lanark, Scotland
Murdoch, D
McFadyen, R
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Glasgow, Glasgow G12 8QQ, Lanark, Scotland
McFadyen, R
McDonagh, T
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Glasgow, Glasgow G12 8QQ, Lanark, Scotland
McDonagh, T
HEART,
2003,
89
: A57
-
A57
[29]
Antihypertensive efficacy, safety and tolerability of the orally active direct renin inhibitor aliskiren added to hydrochlorothiazide (HCTZ) in patients with grade 3 obesity and hypertension
Prescott, Margaret
论文数:
0
引用数:
0
h-index:
0
机构:
Nova Pharmaceut Corp, E Hanover, NJ USA
Prescott, Margaret
Boye, Sam
论文数:
0
引用数:
0
h-index:
0
机构:
Nova Pharmaceut Corp, E Hanover, NJ USA
Boye, Sam
Le Breton, Stephanie
论文数:
0
引用数:
0
h-index:
0
机构:
Nova Pharmaceut Corp, E Hanover, NJ USA
Le Breton, Stephanie
Keefe, Deborah
论文数:
0
引用数:
0
h-index:
0
机构:
Nova Pharmaceut Corp, E Hanover, NJ USA
Keefe, Deborah
Jordan, Jens
论文数:
0
引用数:
0
h-index:
0
机构:
Nova Pharmaceut Corp, E Hanover, NJ USA
Jordan, Jens
INTERNATIONAL JOURNAL OF OBESITY,
2007,
31
: S99
-
S99
[30]
RADIOIMMUNOASSAY FOR CI-992, AN ORALLY-ACTIVE RENIN INHIBITOR
CONNOLLY, CJC
论文数:
0
引用数:
0
h-index:
0
机构:
PARKE DAVIS PHARMACEUT RES,DEPT MED CHEM,ANN ARBOR,MI 48105
CONNOLLY, CJC
HODGES, JC
论文数:
0
引用数:
0
h-index:
0
机构:
PARKE DAVIS PHARMACEUT RES,DEPT MED CHEM,ANN ARBOR,MI 48105
HODGES, JC
KLUTCHKO, SR
论文数:
0
引用数:
0
h-index:
0
机构:
PARKE DAVIS PHARMACEUT RES,DEPT MED CHEM,ANN ARBOR,MI 48105
KLUTCHKO, SR
NORDBLOM, G
论文数:
0
引用数:
0
h-index:
0
机构:
PARKE DAVIS PHARMACEUT RES,DEPT MED CHEM,ANN ARBOR,MI 48105
NORDBLOM, G
BURGER, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
PARKE DAVIS PHARMACEUT RES,DEPT MED CHEM,ANN ARBOR,MI 48105
BURGER, PJ
BARKSDALE, C
论文数:
0
引用数:
0
h-index:
0
机构:
PARKE DAVIS PHARMACEUT RES,DEPT MED CHEM,ANN ARBOR,MI 48105
BARKSDALE, C
MICHNIEWICZ, B
论文数:
0
引用数:
0
h-index:
0
机构:
PARKE DAVIS PHARMACEUT RES,DEPT MED CHEM,ANN ARBOR,MI 48105
MICHNIEWICZ, B
COOK, J
论文数:
0
引用数:
0
h-index:
0
机构:
PARKE DAVIS PHARMACEUT RES,DEPT MED CHEM,ANN ARBOR,MI 48105
COOK, J
TAYLOR, MD
论文数:
0
引用数:
0
h-index:
0
机构:
PARKE DAVIS PHARMACEUT RES,DEPT MED CHEM,ANN ARBOR,MI 48105
TAYLOR, MD
DOHERTY, AM
论文数:
0
引用数:
0
h-index:
0
机构:
PARKE DAVIS PHARMACEUT RES,DEPT MED CHEM,ANN ARBOR,MI 48105
DOHERTY, AM
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY,
1995,
210
: 61
-
MEDI
←
1
2
3
4
5
→