共 17 条
Solidification of meloxicam self-nano emulsifying drug delivery system formulation incorporated into soluble and insoluble carriers using freeze drying method
被引:7
作者:

Kuncahyo, I.
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机构:
Setiabudi Univ, Dept Pharmaceut Sci & Technol, Fac Pharm, Surakarta 57127, Indonesia
Univ Gadjah Mada, Fac Pharm, Sekip Utara 55281, Yogyakarta, Indonesia Setiabudi Univ, Dept Pharmaceut Sci & Technol, Fac Pharm, Surakarta 57127, Indonesia

Choiri, S.
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机构:
Univ Sebelas Maret, Dept Pharm, Ir Sutami 36A, Surakarta 57126, Indonesia Setiabudi Univ, Dept Pharmaceut Sci & Technol, Fac Pharm, Surakarta 57127, Indonesia

Fudholi, A.
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Univ Gadjah Mada, Fac Pharm, Sekip Utara 55281, Yogyakarta, Indonesia Setiabudi Univ, Dept Pharmaceut Sci & Technol, Fac Pharm, Surakarta 57127, Indonesia
机构:
[1] Setiabudi Univ, Dept Pharmaceut Sci & Technol, Fac Pharm, Surakarta 57127, Indonesia
[2] Univ Gadjah Mada, Fac Pharm, Sekip Utara 55281, Yogyakarta, Indonesia
[3] Univ Sebelas Maret, Dept Pharm, Ir Sutami 36A, Surakarta 57126, Indonesia
来源:
INTERNATIONAL CONFERENCE ON ADVANCED MATERIALS FOR BETTER FUTURE 2018
|
2019年
/
578卷
关键词:
IN-VITRO;
NANOEMULSIONS;
OPTIMIZATION;
DESIGN;
SNEDDS;
D O I:
10.1088/1757-899X/578/1/012051
中图分类号:
T [工业技术];
学科分类号:
08 ;
摘要:
Solidification of liquid self-nano emulsifying drug delivery system (SNEDDS) formulation is required to enhance the feasibility and flexibility for further formulation processes. This study purposed to compare the soluble and insoluble carriers namely mannitol and fumed silica, respectively on the nano-emulsion formation and physical properties. The optimized SNEDDS formulation comprising of virgin olive oil, Tween 80, and PEG 400; and meloxicam was impregnated into solid carriers e.g. mannitol and fumed silica using a freeze-drying method. The physical mixture was carried out to compare the aforementioned method. Vibrational spectroscopy, thermal analysis, and morphological characteristic, droplet size and distribution, and drug release were performed to characterize the solid SNEDDS (S-SNEDDS). The result showed that crystallization of meloxicam did not observe in the S-SNEDDS formulations, which confirmed by the vibrational spectroscopy and thermal analysis. The morphological characteristic of S-SNEDDS was similar to the native carriers. The soluble carrier did not affect the formation of the nano-emulsion compared to the insoluble carrier. In addition, the S-SNEDDS enhanced the drug release of meloxicam up to 3-4 folds increment.
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[1]
Formulation of solid self-nanoemulsifying drug delivery systems using N-methyl pyrrolidone as cosolvent
[J].
Agrawal, Anuj G.
;
Kumar, Ashok
;
Gide, Paraag S.
.
DRUG DEVELOPMENT AND INDUSTRIAL PHARMACY,
2015, 41 (04)
:594-604

Agrawal, Anuj G.
论文数: 0 引用数: 0
h-index: 0
机构:
Cachet Pharmaceut Pvt Ltd, Baddi 173205, Solan, India Cachet Pharmaceut Pvt Ltd, Baddi 173205, Solan, India

Kumar, Ashok
论文数: 0 引用数: 0
h-index: 0
机构:
Cachet Pharmaceut Pvt Ltd, Baddi 173205, Solan, India Cachet Pharmaceut Pvt Ltd, Baddi 173205, Solan, India

Gide, Paraag S.
论文数: 0 引用数: 0
h-index: 0
机构:
Dr LH Hiranandani Coll Pharm, Ulhasnagar, Thane, India Cachet Pharmaceut Pvt Ltd, Baddi 173205, Solan, India
[2]
Development and optimization of a meloxicam/-cyclodextrin complex for orally disintegrating tablet using statistical analysis
[J].
Ainurofiq, Ahmad
;
Choiri, Syaiful
.
PHARMACEUTICAL DEVELOPMENT AND TECHNOLOGY,
2018, 23 (05)
:464-475

Ainurofiq, Ahmad
论文数: 0 引用数: 0
h-index: 0
机构:
Sebelas Maret Univ, Dept Pharm, Surakarta, Indonesia Sebelas Maret Univ, Dept Pharm, Surakarta, Indonesia

论文数: 引用数:
h-index:
机构:
[3]
Optimization and characterization of the formation of oil-in-water diazinon nanoemulsions: Modeling and influence of the oil phase, surfactant and sonication
[J].
Badawy, Mohamed E. I.
;
Saad, Abdel-Fattah S. A.
;
Tayeb, El-Sayed H. M.
;
Mohammed, Sondos A.
;
Abd-Elnabi, Amany D.
.
JOURNAL OF ENVIRONMENTAL SCIENCE AND HEALTH PART B-PESTICIDES FOOD CONTAMINANTS AND AGRICULTURAL WASTES,
2017, 52 (12)
:896-911

Badawy, Mohamed E. I.
论文数: 0 引用数: 0
h-index: 0
机构:
Alexandria Univ, Dept Pesticide Chem & Technol, Fac Agr, Alexandria, Egypt Alexandria Univ, Dept Pesticide Chem & Technol, Fac Agr, Alexandria, Egypt

Saad, Abdel-Fattah S. A.
论文数: 0 引用数: 0
h-index: 0
机构:
Alexandria Univ, Fac Agr Saba Basha, Dept Plant Protect, Alexandria, Egypt Alexandria Univ, Dept Pesticide Chem & Technol, Fac Agr, Alexandria, Egypt

Tayeb, El-Sayed H. M.
论文数: 0 引用数: 0
h-index: 0
机构:
Alexandria Univ, Fac Agr Saba Basha, Dept Plant Protect, Alexandria, Egypt Alexandria Univ, Dept Pesticide Chem & Technol, Fac Agr, Alexandria, Egypt

Mohammed, Sondos A.
论文数: 0 引用数: 0
h-index: 0
机构:
Agr Res Ctr, Plant Protect Res Inst, Giza, Egypt Alexandria Univ, Dept Pesticide Chem & Technol, Fac Agr, Alexandria, Egypt

Abd-Elnabi, Amany D.
论文数: 0 引用数: 0
h-index: 0
机构:
Agr Res Ctr, Plant Protect Res Inst, El Nubaria Res Stn, El Nubaria, Egypt Alexandria Univ, Dept Pesticide Chem & Technol, Fac Agr, Alexandria, Egypt
[4]
Study of surfactant combinations and development of a novel nanoemulsion for minimising variations in bioavailability of ezetimibe
[J].
Bali, Vikas
;
Ali, Mushir
;
Ali, Javed
.
COLLOIDS AND SURFACES B-BIOINTERFACES,
2010, 76 (02)
:410-420

Bali, Vikas
论文数: 0 引用数: 0
h-index: 0
机构:
Fac Pharm, Dept Pharmaceut, New Delhi 110062, India Fac Pharm, Dept Pharmaceut, New Delhi 110062, India

Ali, Mushir
论文数: 0 引用数: 0
h-index: 0
机构:
Fac Pharm, Dept Pharmaceut, New Delhi 110062, India Fac Pharm, Dept Pharmaceut, New Delhi 110062, India

Ali, Javed
论文数: 0 引用数: 0
h-index: 0
机构:
Fac Pharm, Dept Pharmaceut, New Delhi 110062, India Fac Pharm, Dept Pharmaceut, New Delhi 110062, India
[5]
Role of solid carriers in pharmaceutical performance of solid supersaturable SEDDS of celecoxib
[J].
Chavan, Rahul B.
;
Modi, Sameer R.
;
Bansal, Arvind K.
.
INTERNATIONAL JOURNAL OF PHARMACEUTICS,
2015, 495 (01)
:374-384

Chavan, Rahul B.
论文数: 0 引用数: 0
h-index: 0
机构:
Natl Inst Pharmaceut Educ & Res, Dept Pharmaceut, Sas Nagar 160062, Punjab, India Natl Inst Pharmaceut Educ & Res, Dept Pharmaceut, Sas Nagar 160062, Punjab, India

Modi, Sameer R.
论文数: 0 引用数: 0
h-index: 0
机构:
Natl Inst Pharmaceut Educ & Res, Dept Pharmaceut, Sas Nagar 160062, Punjab, India Natl Inst Pharmaceut Educ & Res, Dept Pharmaceut, Sas Nagar 160062, Punjab, India

Bansal, Arvind K.
论文数: 0 引用数: 0
h-index: 0
机构:
Natl Inst Pharmaceut Educ & Res, Dept Pharmaceut, Sas Nagar 160062, Punjab, India Natl Inst Pharmaceut Educ & Res, Dept Pharmaceut, Sas Nagar 160062, Punjab, India
[6]
Design and evaluation of self-nanoemulsifying drug delivery systems (SNEDDS) for cefpodoxime proxetil
[J].
Date, Abhijit A.
;
Nagarsenker, M. S.
.
INTERNATIONAL JOURNAL OF PHARMACEUTICS,
2007, 329 (1-2)
:166-172

Date, Abhijit A.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Bombay, Coll Pharm, Dept Pharmaceut, Bombay 400098, Maharashtra, India Univ Bombay, Coll Pharm, Dept Pharmaceut, Bombay 400098, Maharashtra, India

Nagarsenker, M. S.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Bombay, Coll Pharm, Dept Pharmaceut, Bombay 400098, Maharashtra, India Univ Bombay, Coll Pharm, Dept Pharmaceut, Bombay 400098, Maharashtra, India
[7]
Solid self-nanoemulsifying drug delivery systems for oral delivery of polypeptide-k: Formulation, optimization, in-vitro and in-vivo antidiabetic evaluation
[J].
Garg, Varun
;
Kaur, Puneet
;
Singh, Sachin Kumar
;
Kumar, Bimlesh
;
Bawa, Palak
;
Gulati, Monica
;
Yadav, Ankit Kumar
.
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES,
2017, 109
:297-315

Garg, Varun
论文数: 0 引用数: 0
h-index: 0
机构:
Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India

Kaur, Puneet
论文数: 0 引用数: 0
h-index: 0
机构:
Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India

Singh, Sachin Kumar
论文数: 0 引用数: 0
h-index: 0
机构:
Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India

Kumar, Bimlesh
论文数: 0 引用数: 0
h-index: 0
机构:
Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India

Bawa, Palak
论文数: 0 引用数: 0
h-index: 0
机构:
Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India

Gulati, Monica
论文数: 0 引用数: 0
h-index: 0
机构:
Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India

Yadav, Ankit Kumar
论文数: 0 引用数: 0
h-index: 0
机构:
Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India Lovely Profess Univ, Sch Pharmaceut Sci, Phagwara 144411, Punjab, India
[8]
Solid self-nanoemulsifying drug delivery system (S-SNEDDS) of darunavir for improved dissolution and oral bioavailability: In vitro and in vivo evaluation
[J].
Inugala, Spandana
;
Eedara, Basanth Babu
;
Sunkavalli, Sharath
;
Dhurke, Rajeshri
;
Kandadi, Prabhakar
;
Jukanti, Raju
;
Bandari, Suresh
.
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES,
2015, 74
:1-10

Inugala, Spandana
论文数: 0 引用数: 0
h-index: 0
机构:
St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India

Eedara, Basanth Babu
论文数: 0 引用数: 0
h-index: 0
机构:
St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India

Sunkavalli, Sharath
论文数: 0 引用数: 0
h-index: 0
机构:
St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India

Dhurke, Rajeshri
论文数: 0 引用数: 0
h-index: 0
机构:
St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India

Kandadi, Prabhakar
论文数: 0 引用数: 0
h-index: 0
机构:
St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India

Jukanti, Raju
论文数: 0 引用数: 0
h-index: 0
机构:
St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India

Bandari, Suresh
论文数: 0 引用数: 0
h-index: 0
机构:
St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India St Peters Inst Pharmaceut Sci, Dept Pharmaceut, Warangal 506001, Telangana, India
[9]
Improved delivery of poorly soluble compounds using nanoparticle technology: a review
[J].
Kalepu, Sandeep
;
Nekkanti, Vijaykumar
.
DRUG DELIVERY AND TRANSLATIONAL RESEARCH,
2016, 6 (03)
:319-332

Kalepu, Sandeep
论文数: 0 引用数: 0
h-index: 0
机构:
Shri Vishnu Coll Pharm, Dept Pharmaceut Technol, Bhimavaram, Andhra Pradesh, India Shri Vishnu Coll Pharm, Dept Pharmaceut Technol, Bhimavaram, Andhra Pradesh, India

Nekkanti, Vijaykumar
论文数: 0 引用数: 0
h-index: 0
机构:
Western Univ Hlth Sci, Coll Pharm, Pomona, CA USA Shri Vishnu Coll Pharm, Dept Pharmaceut Technol, Bhimavaram, Andhra Pradesh, India
[10]
A novel solid self-nanoemulsifying drug delivery system (S-SNEDDS) for improved stability and oral bioavailability of an oily drug, 1-palmitoyl-2-linoleoyl-3-acetyl-rac-glycerol
[J].
Kim, Kyeong Soo
;
Yang, Eun Su
;
Kim, Dong Shik
;
Kim, Dong Wuk
;
Yoo, Hye Hyun
;
Yong, Chul Soon
;
Youn, Yu Seok
;
Oh, Kyung Taek
;
Jee, Jun-Pil
;
Kim, Jong Oh
;
Jin, Sung Giu
;
Choi, Han Gon
.
DRUG DELIVERY,
2017, 24 (01)
:1018-1025

Kim, Kyeong Soo
论文数: 0 引用数: 0
h-index: 0
机构:
Hanyang Univ, Coll Pharm, Ansan, South Korea
Hanyang Univ, Inst Pharmaceut Sci & Technol, Ansan, South Korea Hanyang Univ, Coll Pharm, Ansan, South Korea

Yang, Eun Su
论文数: 0 引用数: 0
h-index: 0
机构:
Hanyang Univ, Coll Pharm, Ansan, South Korea
Hanyang Univ, Inst Pharmaceut Sci & Technol, Ansan, South Korea Hanyang Univ, Coll Pharm, Ansan, South Korea

Kim, Dong Shik
论文数: 0 引用数: 0
h-index: 0
机构:
Hanyang Univ, Coll Pharm, Ansan, South Korea
Hanyang Univ, Inst Pharmaceut Sci & Technol, Ansan, South Korea Hanyang Univ, Coll Pharm, Ansan, South Korea

Kim, Dong Wuk
论文数: 0 引用数: 0
h-index: 0
机构:
Hanyang Univ, Coll Pharm, Ansan, South Korea
Hanyang Univ, Inst Pharmaceut Sci & Technol, Ansan, South Korea Hanyang Univ, Coll Pharm, Ansan, South Korea

Yoo, Hye Hyun
论文数: 0 引用数: 0
h-index: 0
机构:
Hanyang Univ, Coll Pharm, Ansan, South Korea
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Yong, Chul Soon
论文数: 0 引用数: 0
h-index: 0
机构:
Yeungnam Univ, Coll Pharm, Gyongsan, South Korea Hanyang Univ, Coll Pharm, Ansan, South Korea

Youn, Yu Seok
论文数: 0 引用数: 0
h-index: 0
机构:
Sungkyunkwan Univ, Sch Pharm, Suwon, South Korea Hanyang Univ, Coll Pharm, Ansan, South Korea

Oh, Kyung Taek
论文数: 0 引用数: 0
h-index: 0
机构:
Chung Ang Univ, Coll Pharm, Seoul, South Korea Hanyang Univ, Coll Pharm, Ansan, South Korea

Jee, Jun-Pil
论文数: 0 引用数: 0
h-index: 0
机构:
Chosun Univ, Coll Pharm, Gwangju, South Korea Hanyang Univ, Coll Pharm, Ansan, South Korea

论文数: 引用数:
h-index:
机构:

论文数: 引用数:
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机构:

Choi, Han Gon
论文数: 0 引用数: 0
h-index: 0
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Hanyang Univ, Coll Pharm, Ansan, South Korea
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