Peptidomimetics and Peptide Backbone Modifications

被引：98
作者：
Ahn, Jung-Mo [1 ]
Boyle, Nicholas A. [1 ]
MacDonald, Mary T. [1 ]
Janda, Kim D. [1 ]
机构：
[1] Scripps Res Inst, Dept Chem, La Jolla, CA 92037 USA
来源：
MINI-REVIEWS IN MEDICINAL CHEMISTRY | 2002年 / 2卷 / 05期
关键词：
D O I：
10.2174/1389557023405828
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
The replacement of the amide bond in a peptide backbone is a widely used form of peptide mimicry. Several of the most common amide bond surrogates, including peptidomimetic work done in this laboratory, and their biological applications are presented in this review.
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页码：463 / 473
页数：11
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