Microwave-Promoted Efficient Synthesis of Benzo[h]quinolines by Solvent-Free Three-Component Imino-Diels-Alder Reaction under One-Pot Conditions

被引：17
|
作者：
Sarmah, Manas M. [1 ]
Bhuyan, Debajyoti [1 ]
Prajapati, Dipak [1 ]
机构：
[1] CSIR North East Inst Sci & Technol, Div Med Chem, Jorhat 785006, Assam, India
来源：
SYNLETT | 2013年 / 24卷 / 17期
关键词：
imino-Diels-Alder reaction; metal-catalyzed multicomponent reaction; microwave-assisted organic synthesis; benzo[h]quinolines; SIMPLE ACETANILIDES; REUSABLE CATALYST; ORGANIC-SYNTHESIS; INDIUM TRIFLATE; QUINAZOLINE; CYCLIZATION; QUINOLINE; CAMPTOTHECIN; DERIVATIVES; KETONES;
D O I：
10.1055/s-0033-1339844
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
An one-pot, solvent-free imino Diels-Alder reaction has been developed under microwave conditions using 1-naphthylamine, aldehydes, and electron-deficient terminal alkynes in the presence of a catalytic amount of In(OTf)(3) for construction of benzo[h]quinoline derivatives in short reaction times. The method is clean and operationally simple.
引用
收藏
页码：2245 / 2248
页数：4
相关论文
共 50 条
  • [1] Highly Efficient One-Pot Three-Component Mannich Reaction Under Solvent-Free Conditions
    Azizi, N.
    Ebrahimi, F.
    Saidi, M. R.
    SCIENTIA IRANICA TRANSACTION C-CHEMISTRY AND CHEMICAL ENGINEERING, 2009, 16 (02): : 94 - 98
  • [2] Highly efficient one-pot three-component mannich reaction under solvent-free conditions
    Azizi, N.
    Ebrahimi, F.
    Saidi, M.R.
    Scientia Iranica, 2009, 16 (2 C) : 94 - 98
  • [3] Synthesis of thiohydantoins under one-pot three-component solvent-free conditions
    Song Cao
    Longjie Zhu
    Chuanmeng Zhao
    Xiuhong Tang
    Huajun Sun
    Xin Feng
    Xuhong Qian
    Monatshefte für Chemie - Chemical Monthly, 2008, 139
  • [4] Synthesis of thiohydantoins under one-pot three-component solvent-free conditions
    Cao, Song
    Zhu, Longjie
    Zhao, Chuanmeng
    Tang, Xiuhong
    Sun, Huajun
    Feng, Xin
    Qian, Xuhong
    MONATSHEFTE FUR CHEMIE, 2008, 139 (08): : 923 - 926
  • [5] One-pot three-component reaction for efficient and facile synthesis of γ-nitrocarbonyl compounds under solvent-free conditions
    Chengwei Lü
    Yanhang Liu
    Xiaoxia Zhou
    Jiajing Wang
    Chemical Research in Chinese Universities, 2015, 31 : 208 - 211
  • [6] One-pot Three-component Reaction for Efficient and Facile Synthesis of γ-Nitrocarbonyl Compounds Under Solvent-free Conditions
    Lu Chengwei
    Liu Yanhang
    Zhou Xiaoxia
    Wang Jiajing
    CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 31 (02) : 208 - 211
  • [7] Microwave promoted solvent-free one-pot three-component reaction to 2-pentafluorophenylquinoline derivatives
    Zhang, JM
    Yang, W
    Song, LP
    Cai, M
    Zhu, SZ
    TETRAHEDRON LETTERS, 2004, 45 (29) : 5771 - 5773
  • [8] Microwave-promoted one-pot three-component reaction to [60]Fulleropyrrolidine derivatives
    Zhang, JM
    Yang, W
    Wang, S
    He, P
    Zhu, SH
    SYNTHETIC COMMUNICATIONS, 2005, 35 (01) : 89 - 96
  • [9] One-pot three-component Mannich reaction catalyzed by iodine under solvent-free conditions
    Li Gang
    Long Ruiling
    Yang Jiangli
    Kinetics and Catalysis, 2011, 52
  • [10] One-pot three-component Mannich reaction catalyzed by iodine under solvent-free conditions
    Li Gang
    Long Ruiling
    Yang Jiangli
    KINETICS AND CATALYSIS, 2011, 52 (03) : 397 - 400
12345