Efficient and Easy One-Pot Synthesis of New 3,5-Dioxo-thiazolo[2,3-a] pyrimidine-6-carbonitrile and 4,6-Dioxo-pyrimido[2,1-b][1,3]thiazine-7-carbonitrile Derivatives

被引:10
|
作者
Serrar, H. [1 ]
Boukhris, S. [1 ]
Hassikou, A. [1 ]
Souizi, A. [1 ]
机构
[1] Univ Ibn Tofail, Fac Sci, Lab Synthese Organ Organomet & Theor, Kenitra, Morocco
关键词
ANTIMICROBIAL ACTIVITY; FACILE SYNTHESIS; THIAZOLOPYRIMIDINE; PYRIMIDINE; EPOXIDES; AGENTS;
D O I
10.1002/jhet.2085
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
An easy, fast, and cheap way for the synthesis of the new 3,5-dioxo-thiazolo[2,3-a] pyrimidine-6-carbonitriles and 4,6-dioxo-pyrimido[2,1-b][1,3]thiazine-7-carbonitriles using epoxides alpha-functionalized.
引用
收藏
页码:1269 / 1272
页数:4
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