Zeolite-catalyzed cyclocondensation reaction for the selective synthesis of 3,4-dihydropyrimidin-2(1H)-ones

被引：105

作者：

Rani, VR ^{[1
]}

Srinivas, N ^{[1
]}

Kishan, MR ^{[1
]}

Kulkarni, SJ ^{[1
]}

Raghavan, KV ^{[1
]}

机构：

[1] Indian Inst Chem Technol, Catalysis Div, Hyderabad 7, Andhra Pradesh, India

来源：

GREEN CHEMISTRY | 2001年 / 3卷 / 06期

关键词：

D O I：

10.1039/b107612b

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A zeolite catalyzed, single step and environmentally friendly process for the synthesis of dihydropyrimidinones, a pharmacologically important class of compounds, is reported. Reusability of the catalyst and the ease of separation of pure product, selectively and in high yields in comparison to the classical Biginelli reaction, are a few of the unique features of this process.

引用

页码：305 / 306

页数：2

共 15 条

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