Consecutive Tandem Cycloaddition between Nitriles and Azides; Synthesis of 5-Amino-1H-[1,2,3]-triazoles

被引：15

作者：

Gomes, Ana T. P. C. ^{[1
,2
]}

Martins, Priscila R. C. ^{[2
]}

Rocha, David R. ^{[2
]}

Neves, Maria G. P. M. S. ^{[1
]}

Ferreira, Vitor F. ^{[2
]}

Silva, Artur M. S. ^{[1
]}

Cavaleiro, Jose A. S. ^{[1
]}

da Silva, Fernando de C. ^{[2
]}

机构：

[1] Univ Fed Fluminense, Inst Quim, Dept Quim Organ, BR-24020150 Niteroi, RJ, Brazil

[2] Univ Aveiro, Dept Chem, QOPNA, P-3810193 Aveiro, Portugal

来源：

SYNLETT | 2013年 / 24卷 / 01期

关键词：

triazoles; tandem cycloaddition; consecutive reaction; nitriles; azides; PHARMACOLOGICAL ACTIVITY; INHIBITORY-ACTIVITY; DERIVATIVES; SAR;

D O I：

10.1055/s-0032-1317712

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Novel 5-amino-1H-1,2,3-triazoles were synthesized by a new synthetic route that involves consecutive tandem cycloaddition between nitriles and azides.

引用

页码：41 / 44

页数：4

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