Vicinal diamino functionalities as privileged structural elements in biologically active compounds and exploitation of their synthetic chemistry

被引：374

作者：

Kotti, SRSS ^{[1
]}

Timmons, C ^{[1
]}

Li, GG ^{[1
]}

机构：

[1] Texas Tech Univ, Dept Chem & Biochem, Lubbock, TX 79409 USA

来源：

CHEMICAL BIOLOGY & DRUG DESIGN | 2006年 / 67卷 / 02期

关键词：

imidazolines; vicinal diamines;

D O I：

10.1111/j.1747-0285.2006.00347.x

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

The chemistry, synthetic routes and medicinal properties of vicinal diamines and imidazolines are discussed. Synthetic routes towards chemically and pharmaceutically important molecules containing vicinal diamine functionality are discussed in detail. This mini review article covers the new developments of diamine chemistry between 2000 and 2005.

引用

页码：101 / 114

页数：14

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