共 5 条
[1]
Small Molecule Inhibition of GDC-0449 Refractory Smoothened Mutants and Downstream Mechanisms of Drug Resistance
[J].
Dijkgraaf, Gerrit J. P.
;
Alicke, Bruno
;
Weinmann, Lasse
;
Januario, Thomas
;
West, Kristina
;
Modrusan, Zora
;
Burdick, Dan
;
Goldsmith, Richard
;
Robarge, Kirk
;
Sutherlin, Dan
;
Scales, Suzie J.
;
Gould, Stephen E.
;
Yauch, Robert L.
;
de Sauvage, Frederic J.
.
CANCER RESEARCH,
2011, 71 (02)
:435-444

Dijkgraaf, Gerrit J. P.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

Alicke, Bruno
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

Weinmann, Lasse
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

Januario, Thomas
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

West, Kristina
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

Modrusan, Zora
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

Burdick, Dan
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

Goldsmith, Richard
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

Robarge, Kirk
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

Sutherlin, Dan
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

Scales, Suzie J.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

Gould, Stephen E.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

Yauch, Robert L.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

de Sauvage, Frederic J.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA
[2]
Phase I Trial of Hedgehog Pathway Inhibitor Vismodegib (GDC-0449) in Patients with Refractory, Locally Advanced or Metastatic Solid Tumors
[J].
LoRusso, Patricia M.
;
Rudin, Charles M.
;
Reddy, Josina C.
;
Tibes, Raoul
;
Weiss, Glen J.
;
Borad, Mitesh J.
;
Hann, Christine L.
;
Brahmer, Julie R.
;
Chang, Ilsung
;
Darbonne, Walter C.
;
Graham, Richard A.
;
Zerivitz, Kenn L.
;
Low, Jennifer A.
;
Von Hoff, Daniel D.
.
CLINICAL CANCER RESEARCH,
2011, 17 (08)
:2502-2511

LoRusso, Patricia M.
论文数: 0 引用数: 0
h-index: 0
机构:
Karmanos Canc Inst, Detroit, MI USA Genentech Inc, San Francisco, CA 94080 USA

Rudin, Charles M.
论文数: 0 引用数: 0
h-index: 0
机构:
Johns Hopkins Univ, Baltimore, MD USA Genentech Inc, San Francisco, CA 94080 USA

Reddy, Josina C.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

Tibes, Raoul
论文数: 0 引用数: 0
h-index: 0
机构:
Scottsdale Healthcare, Translat Genom Res Inst TGen, Scottsdale, AZ USA
Scottsdale Healthcare, Virginia G Piper Canc Ctr, Scottsdale, AZ USA Genentech Inc, San Francisco, CA 94080 USA

Weiss, Glen J.
论文数: 0 引用数: 0
h-index: 0
机构:
Scottsdale Healthcare, Translat Genom Res Inst TGen, Scottsdale, AZ USA
Scottsdale Healthcare, Virginia G Piper Canc Ctr, Scottsdale, AZ USA Genentech Inc, San Francisco, CA 94080 USA

Borad, Mitesh J.
论文数: 0 引用数: 0
h-index: 0
机构:
Scottsdale Healthcare, Translat Genom Res Inst TGen, Scottsdale, AZ USA
Scottsdale Healthcare, Virginia G Piper Canc Ctr, Scottsdale, AZ USA Genentech Inc, San Francisco, CA 94080 USA

Hann, Christine L.
论文数: 0 引用数: 0
h-index: 0
机构:
Johns Hopkins Univ, Baltimore, MD USA Genentech Inc, San Francisco, CA 94080 USA

Brahmer, Julie R.
论文数: 0 引用数: 0
h-index: 0
机构:
Johns Hopkins Univ, Baltimore, MD USA Genentech Inc, San Francisco, CA 94080 USA

Chang, Ilsung
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

Darbonne, Walter C.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

Graham, Richard A.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

Zerivitz, Kenn L.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

Low, Jennifer A.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

Von Hoff, Daniel D.
论文数: 0 引用数: 0
h-index: 0
机构:
Scottsdale Healthcare, Translat Genom Res Inst TGen, Scottsdale, AZ USA
Scottsdale Healthcare, Virginia G Piper Canc Ctr, Scottsdale, AZ USA Genentech Inc, San Francisco, CA 94080 USA
[3]
Hedgehog Fights Back: Mechanisms of Acquired Resistance against Smoothened Antagonists
[J].
Metcalfe, Ciara
;
de Sauvage, Frederic J.
.
CANCER RESEARCH,
2011, 71 (15)
:5057-5061

Metcalfe, Ciara
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA

de Sauvage, Frederic J.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA
[4]
Sekulic A, 2012, NEW ENGL J MED, V366, P2171, DOI 10.1056/NEJMoa1113713
[5]
Inhibition of the Hedgehog Pathway in Advanced Basal-Cell Carcinoma.
[J].
Von Hoff, Daniel D.
;
LoRusso, Patricia M.
;
Rudin, Charles M.
;
Reddy, Josina C.
;
Yauch, Robert L.
;
Tibes, Raoul
;
Weiss, Glen J.
;
Borad, Mitesh J.
;
Hann, Christine L.
;
Brahmer, Julie R.
;
Mackey, Howard M.
;
Lum, Bertram L.
;
Darbonne, Walter C.
;
Marsters, James C., Jr.
;
de Sauvage, Frederic J.
;
Low, Jennifer A.
.
NEW ENGLAND JOURNAL OF MEDICINE,
2009, 361 (12)
:1164-1172

Von Hoff, Daniel D.
论文数: 0 引用数: 0
h-index: 0
机构:
Translat Genom Res Inst, Scottsdale, AZ USA
Scottsdale Healthcare, Scottsdale, AZ USA Genentech Inc, San Francisco, CA 94080 USA

LoRusso, Patricia M.
论文数: 0 引用数: 0
h-index: 0
机构:
Karmanos Canc Inst, Detroit, MI USA Genentech Inc, San Francisco, CA 94080 USA

Rudin, Charles M.
论文数: 0 引用数: 0
h-index: 0
机构:
Johns Hopkins Univ, Baltimore, MD USA Genentech Inc, San Francisco, CA 94080 USA

Reddy, Josina C.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

Yauch, Robert L.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

Tibes, Raoul
论文数: 0 引用数: 0
h-index: 0
机构:
Translat Genom Res Inst, Scottsdale, AZ USA
Scottsdale Healthcare, Scottsdale, AZ USA Genentech Inc, San Francisco, CA 94080 USA

Weiss, Glen J.
论文数: 0 引用数: 0
h-index: 0
机构:
Translat Genom Res Inst, Scottsdale, AZ USA
Scottsdale Healthcare, Scottsdale, AZ USA Genentech Inc, San Francisco, CA 94080 USA

Borad, Mitesh J.
论文数: 0 引用数: 0
h-index: 0
机构:
Translat Genom Res Inst, Scottsdale, AZ USA
Scottsdale Healthcare, Scottsdale, AZ USA Genentech Inc, San Francisco, CA 94080 USA

Hann, Christine L.
论文数: 0 引用数: 0
h-index: 0
机构:
Johns Hopkins Univ, Baltimore, MD USA Genentech Inc, San Francisco, CA 94080 USA

Brahmer, Julie R.
论文数: 0 引用数: 0
h-index: 0
机构:
Johns Hopkins Univ, Baltimore, MD USA Genentech Inc, San Francisco, CA 94080 USA

Mackey, Howard M.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

Lum, Bertram L.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

Darbonne, Walter C.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

Marsters, James C., Jr.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

de Sauvage, Frederic J.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA

Low, Jennifer A.
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA