Synthesis, crystal structure and biological activity of a novel anthranilic diamide insecticide containing allyl ether

被引：4

作者：

Zhao, Yu ^{[1
]}

Xiong, Li-xia ^{[1
]}

Xu, Li-ping ^{[1
]}

Wang, Hongxue ^{[1
]}

Xu, Han ^{[1
]}

Li, Hua-bin ^{[1
]}

Tong, Jun ^{[1
]}

Li, Zheng-ming ^{[1
]}

机构：

[1] Nankai Univ, Natl Pesticidal Engn Ctr Tianjin, State Key Lab Elementoorgan Chem, Tianjin 300071, Peoples R China

来源：

RESEARCH ON CHEMICAL INTERMEDIATES | 2013年 / 39卷 / 07期

关键词：

Anthranilic diamide; Ryanodine receptor; Synthesis; Insecticidal activity; FUNGICIDAL ACTIVITY; DFT CALCULATION; 1,2,3-THIADIAZOLE; DERIVATIVES; BIOACTIVITY; POTENT; MOIETY;

D O I：

10.1007/s11164-012-0820-6

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

In search of environmentally benign insecticides with high activity, low toxicity and low residue, a series of novel anthranilic diamides containing allyl ether were designed and synthesized. All the compounds were characterized by H-1 NMR spectroscopy, HRMS or elemental analysis. The single crystal structure of 18e was determined by X-ray diffraction. The insecticidal activities of the new compounds were evaluated. The results showed that some compounds exhibited excellent insecticidal activities against Lepidoptera pests. Among this series compounds, 18l showed 100 % larvicidal activity against Mythimna separate Walker and Plutella xylostella Linnaeus at the test concentration.

引用

页码：3071 / 3088

页数：18

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