CONTIGUOUS GENERATION OF QUATERNARY AND TERTIARY STEREOCENTERS: ONE-POT SYNTHESIS OF CHROMAN-FUSED S-PROLINE-DERIVED CHIRAL OXAZEPINONES

被引：8
作者：
Singh, Ritesh [1 ]
Parai, Maloy Kumar [1 ]
Mondal, Sankalan [1 ]
Panda, Gautam [1 ]
机构：
[1] CSIR, Med & Proc Chem Div, Cent Drug Rearch Inst, Lucknow 226001, Uttar Pradesh, India
来源：
SYNTHETIC COMMUNICATIONS | 2013年 / 43卷 / 02期
关键词：
Chromans; hydrogen peroxide; oxazepinone; alpha; beta-unsaturated amide; COMBINATORIAL LIBRARIES; PRIVILEGED STRUCTURES; DERIVATIVES; CONSTRUCTION; CENTERS;
D O I：
10.1080/00397911.2011.596301
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A new class of chroman-fused S-proline-derived chiral oxazepinones has been synthesized in one pot through contiguous generation of quaternary and tertiary stereocenters.
引用
收藏
页码：253 / 259
页数：7
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