Carbonic anhydrase inhibitors: an editorial

被引：124

作者：

Supuran, Claudiu T. ^{[1
]}

机构：

[1] Univ Firenze, NEUROFARBA Dept, Sect Pharmaceut & Nutriceut Sci, I-50019 Florence, Italy

来源：

EXPERT OPINION ON THERAPEUTIC PATENTS | 2013年 / 23卷 / 06期

关键词：

anticancer; antiglaucoma; anti-obesity; carbonic anhydrase; coumarin; dithiocarbamate; diuretic; inhibitor; polyamine; sulfonamide; SULFONAMIDES; CLONING; POTENT; HONEY;

D O I：

10.1517/13543776.2013.778246

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

This issue of Expert Opinion on Therapeutic Patents is dedicated to carbonic anhydrase (CA, EC 4.2.1.1) inhibitors (CAIs), a highly dynamic research topic in the last years. Several review articles and patent analyses on diuretics and antiglaucoma, antiepileptic, anti-obesity and anticancer agents belonging to the pharmacological class of the CAIs are presented, together with a review on bacterial, fungal and protozoan CAs and their inhibition as a novel means of designing anti-infectives.

引用

页码：677 / 679

页数：3

共 20 条

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